SCHEMBL205064

SCHEMBL205064

COC(=O)c1ccc(C=O)c(Br)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.55
ALDH1A1 P00352 5/20 0.53
ERN1 O75460 6/20 0.53
HTT P42858 2/20 0.50
ALOX15 P16050 1/20 0.50
HCRTR1 O43613 1/20 0.49
HCRTR2 O43614 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
XDH P47989 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
MAPK1 P28482 1/20 0.46
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 2/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22530401 0.90 ALOX15 (0.51) NOTUMALDH1A1ERN1HTTALOX15
SCHEMBL1174813 0.86 ALDH1A1 (0.53) NOTUMALDH1A1ERN1HTTALOX15
SCHEMBL15715947 0.85 NOTUM (0.54) NOTUMALDH1A1ERN1HTTALOX15
SCHEMBL17747083 0.84 ALDH1A1 (0.58) ALDH1A1ERN1HTTALOX15HCRTR1
SCHEMBL15786243 0.83 ALDH1A1 (0.53) ALDH1A1ERN1HTTALOX15HCRTR1
SCHEMBL2989137 0.82 CA12 (0.53) ALDH1A1CA12CA1CA2CA7
SCHEMBL22530239 0.82 KDM4E (0.52) NOTUMALDH1A1HTTALOX15CA12
SCHEMBL30011802 0.82 KDM4E (0.52) NOTUMALDH1A1HTTALOX15CA12
SCHEMBL4808901 0.82 CA12 (0.43) NOTUMALDH1A1ERN1ALOX15CA12
SCHEMBL1134257 0.81 L3MBTL1 (0.51) ALDH1A1ERN1HTTHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4680608-A1 2,6-DIHYDRO-7H-PYRAZOLO[3,4-C]PYRIDIN-7-ONE DERIVATIVES AS ANTI-MALARIAL AGENTS MMV Medicines for Malaria Venture (CH) 2026-01-21 EP disclosed
EP-4081521-B1 SUBSTITUTED TRICYCLIC COMPOUNDS LUPIN LTD (IN) 2025-12-10 EP disclosed
US-20250368667-A1 USP1 INHIBITOR SHANGHAI QILU PHARMACEUTICAL RES AND DEVELOPMENT CENTRE LTD (CN) 2025-12-04 US disclosed
US-12472271-B2 HDAC6 inhibitors and imaging agents THE GENERAL HOSPITAL CORPORATION (US) 2025-11-18 US disclosed
US-20250263405-A1 HISTONE DEACETYLASE 6 INHIBITOR COMPOUNDS AND USES THEREOF VALO HEALTH, INC. 2025-08-21 US disclosed
EP-4582427-A1 USP1 INHIBITOR Shanghai Qilu Pharmaceutical Research and Development Centre Ltd. (CN) 2025-07-09 EP disclosed
CN-119497713-A USP1 inhibitors 上海齐鲁制药研究中心有限公司 2025-02-21 CN disclosed
CN-119462554-A HDAC inhibitor and preparation and application thereof 赛岚(杭州)生物医药科技有限公司 2025-02-18 CN disclosed
EP-4426285-A1 HISTONE DEACETYLASE 6 INHIBITOR COMPOUNDS AND USES THEREOF Valo Health, Inc. (US) 2024-09-11 EP disclosed
EP-4397656-A2 HDAC6 INHIBITORS AND IMAGING AGENTS The General Hospital Corporation (US) 2024-07-10 EP disclosed
EP-2431367-A2 Fused cyclic compounds as GPR40 receptor modulators Takeda Pharmaceutical Company Limited (JP) 2012-03-21 EP disclosed
US-20120046338-A1 FUSED CYCLIC COMPOUNDS YASUMA TSUNEO (JP) 2012-02-23 US disclosed
EP-2041123-B1 FUSED CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2012-02-01 EP disclosed
US-8088821-B2 Fused cyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-01-03 US disclosed
EP-2248812-A2 Fused cyclic compounds as GPR40 receptor modulators Takeda Pharmaceutical Company Limited (JP) 2010-11-10 EP disclosed
US-20100197761-A1 Fused cyclic compounds YASUMA TSUNEO 2010-08-05 US disclosed
US-7732626-B2 Fused cyclic compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed
US-20100004312-A1 FUSED CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-07 US disclosed
EP-2041123-A2 FUSED CYCLIC COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-04-01 EP disclosed
WO-2008001931-A2 FUSED CYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-01-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100004312-A1 FUSED CYCLIC COMPOUNDS GPR119, GLP1R, GPR65 NOTUM 2044/4885ALDH1A1 3122/4885ERN1 2727/4885
US-20250368667-A1 USP1 INHIBITOR USP1, USP2, USP28 NOTUM 3172/4885ALDH1A1 644/4885ERN1 289/4885
US-12472271-B2 HDAC6 inhibitors and imaging agents HDAC1, HDAC6, HDAC11 NOTUM 3049/4885ALDH1A1 2488/4885ERN1 3439/4885
US-20120046338-A1 FUSED CYCLIC COMPOUNDS GPR119, GLP1R, GPR65 NOTUM 2044/4885ALDH1A1 3122/4885ERN1 2727/4885
US-20250263405-A1 HISTONE DEACETYLASE 6 INHIBITOR COMPOUNDS AND USES THEREOF HDAC6, HDAC1, HDAC3 NOTUM 2076/4885ALDH1A1 1144/4885ERN1 3084/4885
US-20100197761-A1 Fused cyclic compounds GPR119, GLP1R, GPR65 NOTUM 2044/4885ALDH1A1 3122/4885ERN1 2727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.