SCHEMBL20729911

SCHEMBL20729911

O=CNCCCC(NC(=O)CNC=O)C(=O)Nc1ccc(CO)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
SIRT1 Q96EB6 6/20 0.36
SIRT2 Q8IXJ6 5/20 0.36
SPHK1 Q9NYA1 1/20 0.36
SIRT5 Q9NXA8 3/20 0.35
BDKRB2 P30411 1/20 0.35
S1PR1 P21453 1/20 0.35
KLKB1 P03952 2/20 0.34
PLG P00747 2/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
F2 P00734 1/20 0.34
PLAU P00749 1/20 0.34
PLAT P00750 1/20 0.34
PRSS1 P07477 1/20 0.34
SIRT3 Q9NTG7 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24788062 0.84 SPHK1 (0.48) SIRT1SPHK1BDKRB2S1PR1KLKB1
SCHEMBL23071786 0.79 SMN1; SMN2 (0.39) LMNASPHK1S1PR1SMN1; SMN2
SCHEMBL20051422 0.77 MEN1 (0.47) LMNAKLKB1PLGF2PLAU
SCHEMBL24728476 0.76 C3AR1 (0.40) SIRT1SIRT2SPHK1SIRT5SIRT3
SCHEMBL20329050 0.76 CA2 (0.42) SIRT5
SCHEMBL25932588 0.76 LTA4H (0.41) SIRT1SIRT2SIRT5KLKB1PLG
SCHEMBL21781895 0.75 SIRT2 (0.33) SIRT1SIRT2SIRT5SIRT3
SCHEMBL24701258 0.74 C3AR1 (0.42) SIRT1SIRT2SIRT5KLKB1PLG
SCHEMBL24539700 0.74 C3AR1 (0.42) SIRT1SIRT2SIRT5KLKB1PLG
SCHEMBL21782008 0.73 CHRNB2 (0.44) SIRT1SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019030284-A1 NEW TARGETED CYTOTOXIC RATJADONE DERIVATIVES AND CONJUGATES THEREOF Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2019-02-14 WO disclosed