SCHEMBL20832016

SCHEMBL20832016

Cc1ccccc1CN1CCN(c2cc(=O)[nH]nc2C)CC1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPC5 Q9UL62 6/20 0.58
KMT2A Q03164 2/20 0.50
LMNA P02545 3/20 0.49
KDM4E B2RXH2 1/20 0.49
HTR7 P34969 2/20 0.47
TNKS O95271 1/20 0.47
PARP1 P09874 1/20 0.47
TNKS2 Q9H2K2 1/20 0.47
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CYP2A13 Q16696 1/20 0.46
ACHE P22303 1/20 0.45
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20831241 0.84 TRPC5 (0.62) TRPC5KDM4EPARP1GAA
SCHEMBL20832014 0.84 TRPC5 (0.53) TRPC5KMT2ALMNAKDM4ETNKS
SCHEMBL20832011 0.76 TRPC5 (0.69) TRPC5KMT2ALMNAKDM4EHTR7
SCHEMBL20831243 0.74 TRPC5 (0.56) TRPC5KMT2AHTR7MEN1HTT
SCHEMBL2923111 0.74 TRPC5 (0.51) TRPC5KMT2ALMNAKDM4ETNKS
SCHEMBL25686925 0.74 TRPC5 (0.61) TRPC5PARP1GAA
SCHEMBL20818113 0.73 TRPC5 (1.00) TRPC5KMT2ATNKSPARP1TNKS2
SCHEMBL20832012 0.73 TRPC5 (0.66) TRPC5PARP1GAA
SCHEMBL20818756 0.72 KMT2A (0.50) TRPC5KMT2ALMNAKDM4ETNKS
SCHEMBL18434116 0.72 ADRB1 (0.42) HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GFB (ABC), LLC 2023-06-29 US disclosed
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF GFB (ABC), LLC 2023-06-29 US disclosed
WO-2019055966-A2 PYRIDAZINONES AND METHODS OF USE THEREOF GOLDFINCH BIO, INC. (US) 2019-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230203028-A1 PYRIDAZINONES AND METHODS OF USE THEREOF PDXK, ATP6V1B1, REN TRPC5 1439/4885KMT2A 3397/4885LMNA 715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.