SCHEMBL2085980

SCHEMBL2085980

COc1ccccc1-c1cccnc1C=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 5/20 0.46
PDE5A O76074 2/20 0.46
AURKA O14965 1/20 0.46
HSD17B10 Q99714 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 1/20 0.44
ERN1 O75460 1/20 0.43
CYP19A1 P11511 1/20 0.42
ALDH1A1 P00352 3/20 0.42
MAOB P27338 1/20 0.42
METAP2 P50579 1/20 0.41
HTR7 P34969 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084338 0.84 NFE2L2 (0.55) NFE2L2NPC1RAB9AERN1
SCHEMBL7608689 0.82 ERN1 (0.47) NFE2L2KDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL8512088 0.82 S100A4 (0.45) KDM4ENPC1TP53GAARAB9A
SCHEMBL27255595 0.80 HTT (0.47) NFE2L2NPC1RAB9ASMN1; SMN2ERN1
SCHEMBL890949 0.80 S100A4 (0.43) KDM4ENPC1TP53GAARAB9A
SCHEMBL11617705 0.78 KMT2A (0.46) HSD17B10KDM4ENPC1TP53RAB9A
SCHEMBL20406217 0.77 POLB (0.50) NFE2L2PDE5AAURKAHSD17B10KDM4E
SCHEMBL4035576 0.77 ALDH1A1 (0.41) NPC1GAAPKMRAB9ASMN1; SMN2
SCHEMBL6065171 0.77 ALDH1A1 (0.53) PDE5AAURKAHSD17B10KDM4ENPC1
SCHEMBL14484609 0.75 CLK4 (0.51) NFE2L2AURKAKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110563641-B Ortho-halogenated phenyl pyridine ketone compound and preparation method thereof 三峡大学 2023-03-24 CN disclosed
EP-1613613-B1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORP (US) 2021-06-02 EP disclosed
CN-110563641-A Ortho-halogenated phenyl pyridine ketone compound and preparation method thereof 三峡大学 2019-12-13 CN disclosed
EP-2010550-B1 POLYMERISATION OF ETHYLENE AND ALPHA-OLEFINS WITH PYRIDINO-IMINOPHENOL COMPLEXES TOTAL RES & TECHNOLOGY FELUY (BE) 2013-06-19 EP disclosed
US-8399582-B2 Polymerisation of ethylene and alpha-olefins with pyridino-iminophenol complexes TOTAL PETROCHEMICALS RESEARCH FELUY (BE) 2013-03-19 US disclosed
US-7863293-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2011-01-04 US disclosed
US-20100160583-A1 Polymerisation of Ethylene and Alpha-Olefins with Pyridino-Iminophenol Complexes TOTAL PETROCHEMICALS RESEARCH FEULY (BE) 2010-06-24 US disclosed
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
US-20080255197-A1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED CORPORATION (CA) 2008-10-16 US disclosed
US-7291631-B2 CXCR4 chemokine receptor binding compounds GENZYME CORPORATION (US) 2007-11-06 US disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed
US-20040209921-A1 CXCR4 chemokine receptor binding comounds ANORMED CORPORATION (CA) 2004-10-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040209921-A1 CXCR4 chemokine receptor binding comounds CXCR4, CXCR1, CXCR3 NFE2L2 1677/4885PDE5A 2364/4885AURKA 4523/4885
US-20080255197-A1 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS CXCR4, CXCR1, CXCR3 NFE2L2 1764/4885PDE5A 1991/4885AURKA 3929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.