SCHEMBL21028150

SCHEMBL21028150

CCc1ccc(S(=O)(=O)NC2(C(N)=O)CC2)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
HSD11B1 P28845 6/20 0.36
FABP4 P15090 6/20 0.35
ADAM17 P78536 1/20 0.35
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
CCR8 P51685 1/20 0.33
CYP2D6 P10635 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16852627 0.84 BRD4 (0.47) BRD4CTSSCTSKHSD11B1FABP4
SCHEMBL15549189 0.82 FABP4 (0.47) BRD4CTSSCTSKHSD11B1FABP4
SCHEMBL18077846 0.82 BRD4 (0.45) BRD4CTSSCTSKHSD11B1FABP4
SCHEMBL21028102 0.81 BRD4 (0.45) BRD4CTSSCTSKHSD11B1FABP4
SCHEMBL15549456 0.76 BRD4 (0.42) BRD4CTSSCTSKHSD11B1
SCHEMBL21028169 0.75 PARG (0.45) BRD4CTSSCTSK
SCHEMBL28122139 0.71 HSD11B1 (0.55) HSD11B1ALDH1A1CYP2D6
SCHEMBL16849173 0.69 CCR8 (0.39) BRD4CTSSCTSKFABP4ALDH1A1
SCHEMBL7791002 0.69 TTR (0.47) ALDH1A1
SCHEMBL28121527 0.68 HSD11B1 (0.46) BRD4CTSSCTSKHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10301272-B2 Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators for the orphan nuclear receptor ROR[γ] PHENEX PHARMACEUTICALS AG (DE) 2019-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10301272-B2 Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators for the orphan nuclear receptor ROR[γ] RORA, RORB, RORC BRD4 982/4885CTSS 4326/4885CTSK 4585/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.