SCHEMBL21101319

SCHEMBL21101319

CN(CCCCN)Cc1nc2ncccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 10/20 0.48
CHRM2 P08172 1/20 0.45
CYP2D6 P10635 1/20 0.45
DRD2 P14416 1/20 0.45
OPRM1 P35372 1/20 0.45
KCNH2 Q12809 1/20 0.45
NUDT1 P36639 1/20 0.43
AURKA O14965 2/20 0.41
CYP2C9 P11712 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
DRD4 P21917 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3936352 0.79 AURKA (0.50) NUDT1AURKACYP2C9NOS1NOS2
Hydrochloric Acid SCHEMBL9396770 0.78 AURKA (0.49) NUDT1AURKACYP2C9NOS1NOS2
SCHEMBL4719992 0.78 NUDT1 (0.53) NUDT1AURKACYP2C9NOS1NOS2
SCHEMBL14131209 0.75 CXCR4 (0.81) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL30096603 0.75 CXCR4 (0.81) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL21101252 0.74 CXCR4 (0.46) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4773954 0.74 NUDT1 (0.59) NUDT1AURKACYP2C9NOS1NOS2
SCHEMBL24823966 0.74 NUDT1 (0.45) NUDT1CYP2C9NOS1NOS2DRD4
SCHEMBL2314765 0.71 DDAH1 (0.55) NUDT1AURKACYP2C9NOS1NOS2
SCHEMBL7002580 0.70 NUDT1 (0.58) NUDT1AURKACYP2C9NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10322111-B2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy GENZYME CORPORATION (US) 2019-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10322111-B2 Chemokine receptor binding heterocyclic compounds with enhanced efficacy CCR5, CXCR4, CXCR3 CXCR4 2/4885CHRM2 2757/4885CYP2D6 3057/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.