SCHEMBL21233332

SCHEMBL21233332

Cc1cc(-c2cncs2)nn1C

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.41
PDE10A Q9Y233 13/20 0.39
CD38 P28907 1/20 0.35
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PIM1 P11309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22952759 0.78 TBXAS1 (0.38) TBXAS1PDE10ACD38ALDH1A1PIM1
SCHEMBL21233171 0.71 ALDH1A1 (0.36) CYP1A2CYP3A4SMN1; SMN2ALDH1A1
SCHEMBL12090639 0.71 ALDH1A1 (0.51) PDE10ACYP1A2CYP3A4SMN1; SMN2ALDH1A1
SCHEMBL15885324 0.70 KEAP1 (0.44) TBXAS1PDE10ACD38
SCHEMBL21233152 0.69 CYP11B2 (0.44) TBXAS1PDE10ACD38CYP11B2SMN1; SMN2
SCHEMBL21233170 0.69 ALDH1A1 (0.37) CYP1A2CYP3A4SMN1; SMN2ALDH1A1
SCHEMBL21233334 0.68 PIM1 (0.37) PDE10ACYP11B1CYP11B2CYP1A2CYP3A4
SCHEMBL21241322 0.68 NMT1 (0.41) CYP11B1CYP11B2CYP1A2CYP3A4SMN1; SMN2
SCHEMBL21233175 0.68 ALDH1A1 (0.33) CYP1A2CYP3A4SMN1; SMN2ALDH1A1
SCHEMBL571374 0.66 HDAC8 (0.50) TBXAS1CD38SMN1; SMN2ALDH1A1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019148851-A1 FIVE-MEMBERED RING-SUBSTITUTED PYRIDAZINOL COMPOUND AND DERIVATIVES THEREOF, PREPARATION METHOD, HERBICIDAL COMPOSITION, AND APPLICATION 青岛清原化合物有限公司 2019-08-08 WO disclosed
WO-2019149260-A1 PYRIDAZINOL COMPOUND, DERIVATIVE THEREOF, PREPARATION METHOD THEREFOR, HERBICIDAL COMPOSITION AND USE THEREOF 青岛清原化合物有限公司 2019-08-08 WO disclosed