SCHEMBL21332907

SCHEMBL21332907

COC(=O)c1nccc2c1nc(Cc1ccccc1)n2C

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RNASEH1 O60930 1/20 0.43
BRD4 O60885 3/20 0.40
CREBBP Q92793 3/20 0.40
EGLN1 Q9GZT9 3/20 0.39
CYP1A2 P05177 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38
DRD2 P14416 1/20 0.38
TBXA2R P21731 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ACSL1 P33121 1/20 0.38
PLA2G2A P14555 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22844069 0.83 L3MBTL1 (0.37) BRD4CREBBPEGLN1L3MBTL1
SCHEMBL21333288 0.79 RXFP1 (0.39) BRD4CREBBPSMN1; SMN2RXFP1TLR7
SCHEMBL9280321 0.77 RNASEH1 (0.48) RNASEH1CYP1A2SMN1; SMN2RXFP1DRD2
SCHEMBL20477374 0.76 RNASEH1 (0.47) RNASEH1CYP1A2SMN1; SMN2RXFP1DRD2
SCHEMBL22079307 0.74 RNASEH1 (0.57) RNASEH1CYP1A2SMN1; SMN2RXFP1L3MBTL1
SCHEMBL21332761 0.74 RXFP1 (0.39) CYP1A2SMN1; SMN2RXFP1TLR7ACSL1
SCHEMBL21333059 0.73 LTA4H (0.51) SMN1; SMN2RXFP1TLR7L3MBTL1
SCHEMBL20477364 0.72 RNASEH1 (0.44) RNASEH1CYP1A2SMN1; SMN2RXFP1DRD2
SCHEMBL20477354 0.71 ADCY10 (0.43) RNASEH1RXFP1DRD2TBXA2RPLA2G2A
SCHEMBL6491001 0.70 PARP1 (0.52) RNASEH1CYP1A2SMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3762377-B1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF UNIV CORNELL (US) 2025-08-20 EP disclosed
US-11964960-B2 Pyridinone- and pyridazinone-based compounds and uses thereof CORNELL UNIVERSITY (US) 2024-04-23 US disclosed
EP-3762377-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF Cook, Timothy, H. (US) 2021-01-13 EP disclosed
US-20200407339-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND USES THEREOF TRI-INSTITUTIONAL THERAPEUTICS DISCOVERY INSTITUTE 2020-12-31 US disclosed
WO-2019173790-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND MEDICAL USES THEREOF HLA TIMOTHY (US) 2019-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200407339-A1 PYRIDINONE- AND PYRIDAZINONE-BASED COMPOUNDS AND USES THEREOF PTGER1, LOXL1, COL1A1 RNASEH1 1523/4885BRD4 2394/4885CREBBP 2747/4885
US-11964960-B2 Pyridinone- and pyridazinone-based compounds and uses thereof PTGER1, LOXL1, COL1A1 RNASEH1 1523/4885BRD4 2394/4885CREBBP 2747/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.