SCHEMBL21342015

SCHEMBL21342015

COc1ccc(C2CN(Cc3ccncc3)C(=O)C[C@H]2NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
FPR1 P21462 4/20 0.42
KMT2A Q03164 1/20 0.42
ALDH1A1 P00352 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPK1 P28482 2/20 0.40
ALOX15 P16050 1/20 0.40
FPR2 P25090 1/20 0.39
LMNA P02545 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
PDE4B Q07343 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21342495 0.89 FPR1 (0.50) KDM1ASMN1; SMN2CYP3A4CYP2C19FPR1
SCHEMBL21342429 0.85 SMN1; SMN2 (0.51) KDM1ASMN1; SMN2FPR1KMT2AALDH1A1
SCHEMBL21342490 0.85 SMN1; SMN2 (0.51) KDM1ASMN1; SMN2FPR1KMT2AALDH1A1
SCHEMBL21342018 0.83 KDM1A (0.47) KDM1ACYP3A4CYP2C19FPR1FPR2
SCHEMBL21342410 0.83 KDM1A (0.47) KDM1ACYP3A4CYP2C19FPR1FPR2
SCHEMBL21342013 0.81 FPR2 (0.59) FPR1FPR2
SCHEMBL21342456 0.80 FPR1 (0.53) KDM1AFPR1ALDH1A1L3MBTL1FPR2
SCHEMBL21342340 0.78 LMNA (0.51) KDM1ASMN1; SMN2KMT2AALDH1A1LMNA
SCHEMBL21342016 0.78 SMN1; SMN2 (0.43) KDM1ASMN1; SMN2CYP3A4CYP2C19KMT2A
SCHEMBL19988732 0.75 FPR1 (0.55) SMN1; SMN2CYP3A4CYP2C19FPR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019170904-A1 PIPERIDINES OR PIPERIDONES SUBSTITUTED WITH UREA AND PHENYL Grünenthal GmbH (DE) 2019-09-12 WO disclosed