SCHEMBL21362568

SCHEMBL21362568

O=C(c1ccc(F)cc1)c1ccc(CC2CC2)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.41
MAPK14 Q16539 2/20 0.39
GRIN2B Q13224 2/20 0.37
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158130 0.82 EPHX2 (0.37) EPHX2HTR2AHTR2C
SCHEMBL20157560 0.81 PTPN1 (0.43)
SCHEMBL20157516 0.80 ALDH1A1 (0.48)
SCHEMBL20157523 0.79 CES2 (0.39)
SCHEMBL20157557 0.78 PTPN1 (0.39) MAPK14
SCHEMBL21351905 0.78 CA2 (0.41)
SCHEMBL11860220 0.77 LTA4H (0.46)
SCHEMBL20157579 0.77 TP53 (0.38)
SCHEMBL20157757 0.77 LMNA (0.50)
SCHEMBL20157552 0.76 LMNA (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed