SCHEMBL21390925

SCHEMBL21390925

CC(C)(CC(=O)CCCc1nc2ccc(OC(F)F)cc2n1C1(C)CCC1)C1CC1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.34
IDH1 O75874 2/20 0.31
HDAC3 O15379 1/20 0.31
PTGS1 P23219 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
ABL1 P00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21390884 0.91 BRD4 (0.33) IDH1HDAC3PTGS1HDAC4HDAC1
SCHEMBL21390928 0.85 HPGDS (0.36) HPGDSIDH1HDAC3PTGS1HDAC4
SCHEMBL21391179 0.85 ACSS2 (0.33) IDH1HDAC3PTGS1HDAC4HDAC1
SCHEMBL21391117 0.83 POLB (0.31)
SCHEMBL21390820 0.83 ACSS2 (0.33) IDH1HDAC3HDAC4HDAC1HDAC2
SCHEMBL21390678 0.82 TRPV4 (0.32)
SCHEMBL21354758 0.80 HPGDS (0.37) HPGDSIDH1ABL1
SCHEMBL21391182 0.78 PDE2A (0.31)
SCHEMBL21391003 0.78
SCHEMBL21391016 0.77 HDAC1 (0.36) HPGDSIDH1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed