SCHEMBL21399403

SCHEMBL21399403

CN(C(N)=O)c1ccc(OCCN)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.46
POLB P06746 1/20 0.46
TAAR1 Q96RJ0 1/20 0.44
LTA4H P09960 2/20 0.43
PLA2G2A P14555 1/20 0.43
HDAC1 Q13547 1/20 0.42
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
MCHR1 Q99705 2/20 0.41
CYP19A1 P11511 2/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
CYP3A4 P08684 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006543 0.83 PARP10 (0.58) SMN1; SMN2POLBALDH1A1LMNAMAPT
SCHEMBL6711589 0.80 TAAR1 (0.44) SMN1; SMN2TAAR1LTA4HPLA2G2ACYP19A1
SCHEMBL7615944 0.77 CA1 (0.53) SMN1; SMN2ALDH1A1MAPTESR2
SCHEMBL7996955 0.76 LMNA (0.49) SMN1; SMN2LTA4HALDH1A1LMNAMAPT
SCHEMBL10754241 0.75 ALDH1A1 (0.59) SMN1; SMN2TAAR1ALDH1A1MAPTCYP19A1
Hydrochloric Acid SCHEMBL12503056 0.73 ALDH1A1 (0.58) SMN1; SMN2ALDH1A1MAPTCYP19A1ESR1
SCHEMBL6122034 0.73 PARP10 (0.70) TAAR1ALDH1A1CYP19A1ESR1ESR2
SCHEMBL6714503 0.73 TAAR1 (0.75) SMN1; SMN2TAAR1LTA4HPLA2G2AALDH1A1
SCHEMBL27321565 0.73 LOXL2 (0.44) SMN1; SMN2KEAP1NFE2L2
SCHEMBL926743 0.72 ALOX5 (0.50) SMN1; SMN2LTA4HKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019182942-A1 TYROSINE-SPECIFIC FUNCTIONALIZED INSULIN AND INSULIN ANALOGS MERCK SHARP & DOHME CORP. (US) 2019-09-26 WO disclosed