Phosphoric Acid

Phosphoric Acid

SCHEMBL21465129

Nc1ncnc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1I.O=P(O)(O)O.O=P(O)(O)O.O=P(O)(O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Phosphoric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 known ✓ P27487 1/20 0.72
ADRB2 known ✓ P07550 1/20 0.62
KCNH2 known ✓ Q12809 1/20 0.62
ADORA3 P0DMS8 4/20 0.72
ADORA1 P30542 3/20 0.72
SMN1; SMN2 Q16637 3/20 0.72
MEN1 O00255 1/20 0.72
SLC28A1 O00337 1/20 0.72
MAP3K7 O43318 1/20 0.72
SLC28A2 O43868 1/20 0.72
GAPDH P04406 1/20 0.72
MAPK1 P28482 1/20 0.72
ADORA2A P29274 1/20 0.72
ADORA2B P29275 1/20 0.72
STAT6 P42226 1/20 0.72
PI4KA P42356 1/20 0.72
KMT2A Q03164 1/20 0.72
PI4K2B Q8TCG2 1/20 0.72
DOT1L Q8TEK3 1/20 0.72
SLC29A1 Q99808 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16341965 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL15798533 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL14946319 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL4463227 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL4463234 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL4463230 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL14853733 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
SCHEMBL31388262 0.94 ADORA3 (0.80) ADORA3ADORA1SMN1; SMN2DPP4MEN1
Adenosine SCHEMBL468212 0.90 ADORA1 (0.89) ADORA3ADORA1SMN1; SMN2DPP4MEN1
Adenosine SCHEMBL1746637 0.90 ADORA1 (0.89) ADORA3ADORA1SMN1; SMN2DPP4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230242569-A1 PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE 2023-08-03 US disclosed
US-20230212204-A1 REAGENTS AND THEIR USE FOR MODULAR ENANTIODIVERGENT SYNTHESIS OF C-P BONDS THE SCRIPPS RESEARCH INSTITUTE 2023-07-06 US disclosed
US-11613554-B2 Phosphorous (V)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (V) compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2023-03-28 US disclosed
WO-2021146391-A1 REAGENTS AND THEIR USE FOR MODULAR ENANTIODIVERGENT SYNTHESIS OF C–P BONDS BRISTOL-MYERS SQUIBB COMPANY (US) 2021-07-22 WO disclosed
EP-3774824-A1 NOVEL PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS Bristol-Myers Squibb Company (US) 2021-02-17 EP disclosed
US-20190322694-A1 NOVEL PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE 2019-10-24 US disclosed
WO-2019200273-A1 NOVEL PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2019-10-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242569-A1 PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS PPIP5K2, INPP5B, PTMS DPP4 562/4885ADRB2 4850/4885KCNH2 2017/4885
US-11613554-B2 Phosphorous (V)-based reagents, processes for the preparation thereof, and their use in making stereo-defined organophoshorous (V) compounds PPIP5K2, INPP5B, PTMS DPP4 562/4885ADRB2 4850/4885KCNH2 2017/4885
US-20190322694-A1 NOVEL PHOSPHOROUS (V)-BASED REAGENTS, PROCESSES FOR THE PREPARATION THEREOF, AND THEIR USE IN MAKING STEREO-DEFINED ORGANOPHOSHOROUS (V) COMPOUNDS PPIP5K2, INPP5B, PTMS DPP4 590/4885ADRB2 4849/4885KCNH2 2307/4885
US-20230212204-A1 REAGENTS AND THEIR USE FOR MODULAR ENANTIODIVERGENT SYNTHESIS OF C-P BONDS PNKP, POLL, RNGTT DPP4 2451/4885ADRB2 4399/4885KCNH2 3699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.