SCHEMBL21697537

SCHEMBL21697537

OC(c1cc2ccccc2s1)c1cc(Br)c(OCc2ccccc2)cc1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 4/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36
F9 P00740 1/20 0.36
F10 P00742 1/20 0.36
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PTGER1 P34995 1/20 0.35
SCD O00767 1/20 0.35
PTGES O14684 1/20 0.34
ALOX5 P09917 1/20 0.34
PSEN1 P49768 1/20 0.34
S1PR1 P21453 2/20 0.33
DRD1 P21728 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21697612 0.85 SMN1; SMN2 (0.37) F9F10RAB9ASMN1; SMN2DRD1
SCHEMBL16020910 0.85 PTGES (0.35) RAB9APTGESALOX5PSEN1S1PR1
SCHEMBL20741824 0.84 ABCB1 (0.41) RAB9ASMN1; SMN2DRD1SLC6A2SLC6A4
SCHEMBL21697645 0.82 HTR2A (0.37) MRGPRX4F9F10RAB9ASMN1; SMN2
SCHEMBL16018672 0.78 ALOX5 (0.36) PTGESALOX5
SCHEMBL21697564 0.77 FFAR1 (0.37) MRGPRX4F9F10RAB9ASMN1; SMN2
SCHEMBL21697652 0.77 THRB (0.38) SMN1; SMN2DRD1SLC6A2SLC6A4SLC6A3
SCHEMBL21697575 0.76 THRB (0.38) SMN1; SMN2
SCHEMBL21697589 0.75 PTGER1 (0.37) MRGPRX4RAB9ASMN1; SMN2PTGER1
SCHEMBL16020940 0.72 RAB9A (0.34) RAB9APTGESALOX5SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968258-B1 DUAL SGLT1/SGLT2 INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2020-02-12 EP disclosed