SCHEMBL2170413

SCHEMBL2170413

Nc1cc(NS(=O)(=O)c2ccccc2)ccc1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 3/20 0.63
KEAP1 Q14145 2/20 0.60
MAPT P10636 2/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HTR6 P50406 2/20 0.59
ALDH1A1 P00352 3/20 0.59
LMNA P02545 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
KMT2A Q03164 4/20 0.56
PKM P14618 3/20 0.56
MEN1 O00255 3/20 0.56
IL1RN P18510 1/20 0.55
ERAP1 Q9NZ08 1/20 0.55
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
GAA P10253 2/20 0.53
GFER P55789 1/20 0.53
APOBEC3G Q9HC16 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8589428 0.85 FFAR4 (0.73) FFAR4KEAP1MAPTHTR6ALDH1A1
SCHEMBL5163794 0.85 LMNA (0.62) FFAR4KEAP1MAPTHTR6ALDH1A1
SCHEMBL3320242 0.84 MAPT (0.73) KEAP1MAPTNPSR1HTR6ALDH1A1
SCHEMBL3780986 0.82 GAA (0.67) FFAR4KEAP1MAPTHTR6ALDH1A1
SCHEMBL5484585 0.81 ALDH1A1 (0.74) MAPTNPSR1ALDH1A1LMNAKMT2A
SCHEMBL17557163 0.81 FFAR4 (0.63) FFAR4KEAP1MAPTHTR6ALDH1A1
SCHEMBL7572838 0.81 PKM (0.67) FFAR4KEAP1HTR6ALDH1A1LMNA
SCHEMBL8016507 0.81 GAA (0.69) FFAR4KEAP1NPSR1HTR6ALDH1A1
SCHEMBL16041517 0.81 LMNA (0.57) FFAR4KEAP1MAPTHTR6ALDH1A1
SCHEMBL3930917 0.81 FFAR4 (0.68) FFAR4KEAP1HTR6ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346847-B1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LTD (IN) 2013-05-15 EP disclosed
US-8404720-B2 Aryl sulfonamide amine compounds and their use as 5-HT6 ligands SUVEN LIFE SCIENCES LIMITED (IN) 2013-03-26 US disclosed
US-20120129816-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2012-05-24 US disclosed
CN-102159564-A Arylsulfonamide compounds and their use as 5-HT6 ligands SUVEN LIFE SCIENCES LTD 2011-08-17 CN disclosed
EP-2346847-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS Suven Life Sciences Limited (IN) 2011-07-27 EP disclosed
WO-2010032258-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS SUVEN LIFE SCIENCES LIMITED (IN) 2010-03-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120129816-A1 ARYL SULFONAMIDE AMINE COMPOUNDS AND THEIR USE AS 5-HT6 LIGANDS HTR6, HTR1A, HTR5A FFAR4 217/4885KEAP1 3660/4885MAPT 69/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.