SCHEMBL2170780

SCHEMBL2170780

CC(C)C(=O)NC(=O)C(C)C(c1cn[nH]c1)c1ncccn1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
NOS2 P35228 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
CDK5 Q00535 1/20 0.31
NPC1 O15118 1/20 0.30
TP53 P04637 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170615 0.86 ROCK2 (0.34) CYP2C8CYP2D6CYP2C9CYP2C19NOS2
SCHEMBL2169013 0.75 RIPK1 (0.31) CYP2C8CYP2D6CYP2C9CYP2C19
SCHEMBL2170749 0.66 NOS2 (0.33) ALDH1A1NOS2
SCHEMBL2170787 0.64 NOS2 (0.39) ALDH1A1LMNAKDM4EHTTNOS2
SCHEMBL2169288 0.63 CYP2C19 (0.34) LMNACYP2D6CYP2C19NOS2RAB9A
SCHEMBL13373478 0.62 KMT2A (0.47) ALDH1A1KDM4EHTTNOS2CCNE1
SCHEMBL509533 0.61 NOS2 (0.42) ALDH1A1LMNAKDM4ECYP2C9NOS2
SCHEMBL15742821 0.60 HRH2 (0.43) ALDH1A1CYP2D6CYP2C19NOS2
SCHEMBL2583496 0.60 NOS2 (0.45) LMNANOS2
SCHEMBL1236387 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130281455-A1 Phenylpyri(mi)dinylazoles BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-10-24 US disclosed
US-20110183978-A1 Phenylpyri(mi)dinylazoles BAYER CROPSCIENCE AG (DE) 2011-07-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130281455-A1 Phenylpyri(mi)dinylazoles PIR, PIN4, PNN ALDH1A1 516/4885LMNA 2389/4885KDM4E 2314/4885
US-20110183978-A1 Phenylpyri(mi)dinylazoles PIR, PIN4, PNN ALDH1A1 516/4885LMNA 2389/4885KDM4E 2314/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.