SCHEMBL21708773

SCHEMBL21708773

CCCC(F)OC(=O)C(C)(CN)c1c(F)cccc1F

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.33
TAS1R1 Q7RTX1 2/20 0.33
PRSS1 P07477 1/20 0.32
CTSG P08311 1/20 0.32
CTRB1 P17538 1/20 0.32
CMA1 P23946 1/20 0.32
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708708 0.92 SMN1; SMN2 (0.33) TAS1R3TAS1R1ALDH1A1
SCHEMBL21708674 0.79 ADRB2 (0.33) TAS1R3TAS1R1PRSS1CTSGCTRB1
SCHEMBL21708655 0.77 MEN1 (0.38) TAS1R3TAS1R1PRSS1CTSGCTRB1
SCHEMBL21656189 0.76 CTSS (0.33)
SCHEMBL21708725 0.76 SMN1; SMN2 (0.35) ALDH1A1HPGD
SCHEMBL21708656 0.76 TAS1R3 (0.35) TAS1R3TAS1R1
SCHEMBL21708779 0.74 NPC1 (0.33) TAS1R3TAS1R1ALDH1A1HPGD
SCHEMBL21708691 0.74 LMNA (0.36) ADRB2ADRB1ADRB3ALDH1A1
SCHEMBL21631960 0.73 PTGFR (0.38)
SCHEMBL21708652 0.72 TAS1R3 (0.34) TAS1R3TAS1R1PRSS1CTSGCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed