SCHEMBL21758196

SCHEMBL21758196

O=C(O)C(Cl)(Cl)c1cccc2c1Cc1ccccc1-2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
HTR2B P41595 4/20 0.43
HTR7 P34969 2/20 0.43
PNMT P11086 1/20 0.41
HSP90AA1 P07900 2/20 0.41
SRD5A2 P31213 2/20 0.41
CYP1A2 P05177 3/20 0.38
BCHE P06276 2/20 0.37
ACHE P22303 1/20 0.37
GSR P00390 1/20 0.37
DRD2 P14416 2/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
HTR2C P28335 2/20 0.35
ADRA1D P25100 1/20 0.35
HTR2A P28223 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
MAOA P21397 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28668245 0.84 NPC1 (0.49) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL30996992 0.84 NPC1 (0.49) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL1539672 0.77 PNMT (0.46) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL8971039 0.77 PNMT (0.46) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL2938536 0.75 RAB9A (0.47) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL2687014 0.74 PNMT (0.44) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL7877087 0.73 PNMT (0.49) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL5837265 0.73 PNMT (0.49) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL2043313 0.73 PNMT (0.49) NPC1RAB9AHTR2BHTR7PNMT
SCHEMBL27942181 0.73 PNMT (0.49) NPC1RAB9AHTR2BHTR7PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11884619-B2 Reagents and methods for esterification WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2024-01-30 US disclosed
US-20220055979-A1 Reagents and Methods for Esterification WISCONSIN ALUMNI RESEARCH FOUNDATION 2022-02-24 US disclosed
US-11091423-B2 Reagents and methods for esterification WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2021-08-17 US disclosed
US-20200190011-A1 Reagents and Methods for Esterification WISCONSIN ALUMNI RESEARCH FOUNDATION 2020-06-18 US disclosed
US-10577303-B1 Reagents and methods for esterification WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2020-03-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200190011-A1 Reagents and Methods for Esterification ADCY1, ADCY4, ADCY7 NPC1 3038/4885RAB9A 1875/4885HTR2B 2398/4885
US-11091423-B2 Reagents and methods for esterification ADCY1, ADCY4, ADCY7 NPC1 3038/4885RAB9A 1875/4885HTR2B 2398/4885
US-10577303-B1 Reagents and methods for esterification ADCY1, ADCY4, ADCY7 NPC1 3038/4885RAB9A 1875/4885HTR2B 2398/4885
US-11884619-B2 Reagents and methods for esterification ADCY1, ADCY4, ADCY7 NPC1 3038/4885RAB9A 1875/4885HTR2B 2398/4885
US-20220055979-A1 Reagents and Methods for Esterification ADCY1, ADCY4, ADCY7 NPC1 3038/4885RAB9A 1875/4885HTR2B 2398/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.