SCHEMBL21795663

SCHEMBL21795663

NC(=O)OC1CCOCC1COc1ccc(-c2ccc(F)cn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.39
GRM5 P41594 3/20 0.38
HDAC1 Q13547 2/20 0.37
HDAC2 Q92769 2/20 0.37
GRIA2 P42262 1/20 0.37
GPR119 Q8TDV5 1/20 0.35
FPR2 P25090 2/20 0.34
SCN9A Q15858 2/20 0.34
NPC1 O15118 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
GRM4 Q14833 2/20 0.34
FFAR4 Q5NUL3 4/20 0.33
AXL P30530 1/20 0.33
MERTK Q12866 1/20 0.33
DGAT1 O75907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21795648 0.88 XDH (0.39) XDHGPR119GRM4FFAR4DGAT1
SCHEMBL21795636 0.88 XDH (0.39) XDHGPR119GRM4FFAR4DGAT1
SCHEMBL21795638 0.87 KDM4E (0.42) XDHGPR119SCN9A
SCHEMBL12986558 0.87 GRM5 (0.38) GRM5SCN9AGRM4FFAR4AXL
SCHEMBL15420322 0.80 GRM5 (0.41) XDHGRM5HDAC1HDAC2GRIA2
SCHEMBL21795659 0.80 NPC1 (0.39) XDHGPR119NPC1FFAR4
SCHEMBL21795667 0.78 FFAR4 (0.37) GRM4FFAR4DGAT1
SCHEMBL21795670 0.78 KCNH2 (0.35) GPR119GRM4FFAR4DGAT1
SCHEMBL21795654 0.77 GRM5 (0.37) XDHGRM5FPR2SCN9AGRM4
SCHEMBL21795640 0.77 PARP15 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694472-B1 SULFONAMIDE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2020-03-11 EP disclosed