SCHEMBL21798490

SCHEMBL21798490

C[C@H](c1ccccc1)N(CCCc1ccccc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
CHRM1 P11229 1/20 0.49
DRD1 P21728 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A4 P31645 1/20 0.49
ADRA1A P35348 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KCNH2 Q12809 1/20 0.49
KMT2A Q03164 3/20 0.48
SIGMAR1 Q99720 2/20 0.48
MEN1 O00255 2/20 0.48
EPHX2 P34913 2/20 0.47
ALOX5 P09917 1/20 0.46
AGTR2 P50052 1/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21798493 1.00 CHRM2 (0.49) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL22327659 0.82 L3MBTL1 (0.43) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL28032109 0.80 ALOX5 (0.47) OPRM1KMT2AMEN1ALOX5KDM4E
SCHEMBL21798476 0.79 CYP2C19 (0.41) OPRM1KMT2AMEN1ALOX5CYP2C19
SCHEMBL21798479 0.79 CYP2C19 (0.41) OPRM1KMT2AMEN1ALOX5CYP2C19
SCHEMBL14865109 0.78 MEN1 (0.40) SLC6A2SLC6A4SLC6A3KMT2AMEN1
SCHEMBL12767573 0.78 OPRM1 (0.48) CHRM2HTR1AADRA2ACHRM1DRD1
SCHEMBL7381782 0.78 HPGD (0.47) KMT2ASIGMAR1MEN1ALOX5CYP2D6
SCHEMBL960788 0.78 ALOX5 (0.45) OPRM1KMT2AMEN1ALOX5
SCHEMBL2479871 0.76 ALOX5 (0.50) ADRA2AOPRM1KCNH2KMT2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10738064-B2 Chiral α-amino tertiary boronic esters PURDUE RESEARCH FOUNDATION (US) 2020-08-11 US disclosed
US-20200079799-A1 Novel Chiral Alfa-Amino Tertiary Boronic Esters PURDUE RESEARCH FOUNDATION (US) 2020-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200079799-A1 Novel Chiral Alfa-Amino Tertiary Boronic Esters HBB, BCAT1, BCAT2 CHRM2 4390/4885HTR1A 4152/4885ADRA2A 1234/4885
US-10738064-B2 Chiral α-amino tertiary boronic esters HBB, BCAT1, BCAT2 CHRM2 4263/4885HTR1A 2868/4885ADRA2A 895/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.