SCHEMBL22015593

SCHEMBL22015593

CC(=O)Cc1c(C(C)C)cc(F)c(F)c1C(C)C

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.32
EIF4A3 P38919 2/20 0.31
GCGR P47871 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19475213 0.87 EIF4A3 (0.36) NLRP3EIF4A3GCGRGAA
SCHEMBL20698765 0.86 SIRT1 (0.35) NLRP3EIF4A3GCGR
SCHEMBL19507330 0.83 MTNR1A (0.40) NLRP3GAA
SCHEMBL22014723 0.79 GABRA1 (0.35) EIF4A3
SCHEMBL23692140 0.79
SCHEMBL22014897 0.78 NLRP3 (0.41) NLRP3EIF4A3GCGRGAA
SCHEMBL27110079 0.77 CA1 (0.41)
SCHEMBL19621872 0.73 CA1 (0.46) NLRP3GAA
SCHEMBL15082628 0.70 GABRA1 (0.31)
SCHEMBL22014632 0.70 MTNR1A (0.37) NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020102574-A1 THE COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RESEARCH, INC. (US) 2020-05-22 WO disclosed