SCHEMBL221237

SCHEMBL221237

O=C1c2ccccc2C(=O)N1CCS(=O)(=O)NC1CCN(C2CC2)CC1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.42
KDM1A O60341 1/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 2/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
DRD2 P14416 2/20 0.39
HPGD P15428 2/20 0.39
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL222333 0.83 MAOB (0.52) ACHEKDM1AALDH1A1DRD2
SCHEMBL219755 0.80 HTR1A (0.42) ACHEKDM1AALDH1A1TSHR
SCHEMBL19739574 0.77 HPGD (0.56) ACHEALDH1A1MAPK1HPGD
SCHEMBL4457921 0.75 HPGD (0.60) ACHEALDH1A1MAPK1DRD2HPGD
SCHEMBL16528120 0.75 MAPK1 (0.46) ACHEALDH1A1MAPK1HTTHPGD
SCHEMBL220470 0.70 SMYD3 (0.38) ALDH1A1DRD2ADRA1DADRA1AADRA1B
SCHEMBL3757316 0.70 GLS (0.49)
Tert-Butyl Formate SCHEMBL27733639 0.70 ACHE (0.40) ACHEALDH1A1MAPK1TSHRDRD2
SCHEMBL3759156 0.69 CASP3 (0.49) ALDH1A1HPGD
SCHEMBL221548 0.69 BRD4 (0.57) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088925-B2 low molecular weight factor Xa specific blood clotting inhibitors; less side effects; 5-Chloro-thiophene-2-carboxylic acid [2-(1-isopropyl-piperidin-4-ylsulfamoyl)-ethyl]-amide; thromboembolic diseases or restenosis; antithrombotic agents SANOFI-AVENTIS (FR) 2012-01-03 US disclosed