SCHEMBL22202029

SCHEMBL22202029

CC1(C)CB(c2ccc3c(c2)CCN3)OC1(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HRH3 Q9Y5N1 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
KDM4E B2RXH2 2/20 0.31
MAPT P10636 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
GAA P10253 1/20 0.31
THRB P10828 1/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
HTT P42858 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12470951 0.80 DRD2 (0.45) DRD2DRD4CA1CA2CA9
SCHEMBL19003095 0.77 CYP11B1 (0.30) SMN1; SMN2CA12CA1CA2KDM4E
SCHEMBL24135395 0.72 CASP1 (0.41) HRH3CASP1CASP7HSD17B10
SCHEMBL21382549 0.71 KDM4E (0.43) DRD2DRD4HRH3CA12CA1
SCHEMBL21433623 0.69 ALDH1A1 (0.41) DRD2SMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL24094424 0.69
SCHEMBL24820904 0.68 LPL (0.40) DRD2DRD4SMN1; SMN2CA12CA1
SCHEMBL19981776 0.68 LPL (0.33)
SCHEMBL21154235 0.67 LPL (0.49)
SCHEMBL12031006 0.67 LPL (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020142486-A1 KINASE INHIBITOR COMPOUNDS AND COMPOSITIONS AND METHODS OF USE ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2020-07-09 WO disclosed