SCHEMBL2234091

SCHEMBL2234091

O/C(=C(/O)c1ccccn1)c1ccccn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.65
L3MBTL1 Q9Y468 2/20 0.65
P4HTM Q9NXG6 2/20 0.65
NAPRT Q6XQN6 1/20 0.65
CES2 O00748 1/20 0.61
CES1 P23141 1/20 0.61
KMT2A Q03164 4/20 0.58
ALDH1A1 P00352 5/20 0.56
KDM4E B2RXH2 7/20 0.52
NPC1 O15118 4/20 0.52
RAB9A P51151 4/20 0.52
MAPT P10636 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
NPSR1 Q6W5P4 2/20 0.52
CCR6 P51684 1/20 0.52
GSK3B P49841 1/20 0.50
PKM P14618 3/20 0.48
POLB P06746 2/20 0.47
GAA P10253 2/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141120 1.00 LMNA (0.65) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL23340688 1.00 LMNA (0.65) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL18219728 0.85 ALDH1A1 (0.59) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL25983246 0.85 LMNA (0.50) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL13225623 0.84 KMT2A (0.59) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL5642554 0.83
SCHEMBL5610095 0.80 CES2 (0.69) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL5610101 0.80 CES2 (0.69) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL28465997 0.80 CES2 (0.64) LMNAL3MBTL1P4HTMNAPRTCES2
SCHEMBL2489302 0.80 CES2 (0.64) LMNAL3MBTL1P4HTMNAPRTCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10017474-B1 Method of synthesizing (E)-1,2-di(pyridin-2-yl) ethene-1,2-diol KING SAUD UNIVERSITY (SA) 2018-07-10 US claimed
EP-2025697-B1 Process to obtain dimers, trimers and up to polymers from pyridinemethanol derivatives compounds BENEMERITA UNIVERSIDAD AUTONOMA DE PUEBLA (MX) 2013-12-18 EP claimed
US-20090043063-A1 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds PERCINO ZACARIAS, Maria Judith (MX) 2009-02-12 US claimed
US-11718607-B2 Atypical coupling method for the preparation of 1,2-di(thiophen-2-yl)ethene-1,2-diol compounds via a Cu(II) catalyst QATAR UNIVERSITY (QA) 2023-08-08 US disclosed
US-11718607-B2 Atypical coupling method for the preparation of 1,2-di(thiophen-2-yl)ethene-1,2-diol compounds via a Cu(II) catalyst QATAR UNIVERSITY (QA) 2023-08-08 US disclosed
US-11718607-B2 Atypical coupling method for the preparation of 1,2-di(thiophen-2-yl)ethene-1,2-diol compounds via a Cu(II) catalyst QATAR UNIVERSITY (QA) 2023-08-08 US disclosed
US-20220204487-A1 ATYPICAL COUPLING METHOD FOR THE PREPARATION OF 1,2-DI(THIOPHEN-2-YL)ETHENE-1,2-DIOL COMPOUNDS VIA A CU(II) CATALYST QATAR UNIVERSITY (QA) 2022-06-30 US disclosed
US-20220204487-A1 ATYPICAL COUPLING METHOD FOR THE PREPARATION OF 1,2-DI(THIOPHEN-2-YL)ETHENE-1,2-DIOL COMPOUNDS VIA A CU(II) CATALYST QATAR UNIVERSITY (QA) 2022-06-30 US disclosed
US-10017474-B1 Method of synthesizing (E)-1,2-di(pyridin-2-yl) ethene-1,2-diol KING SAUD UNIVERSITY (SA) 2018-07-10 US disclosed
US-10017474-B1 Method of synthesizing (E)-1,2-di(pyridin-2-yl) ethene-1,2-diol KING SAUD UNIVERSITY (SA) 2018-07-10 US disclosed
US-10017474-B1 Method of synthesizing (E)-1,2-di(pyridin-2-yl) ethene-1,2-diol KING SAUD UNIVERSITY (SA) 2018-07-10 US disclosed
EP-2025697-B1 Process to obtain dimers, trimers and up to polymers from pyridinemethanol derivatives compounds BENEMERITA UNIVERSIDAD AUTONOMA DE PUEBLA (MX) 2013-12-18 EP disclosed
US-7989583-B2 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds BENEMERITA UNIVERSIDAD AUTONOMA DE PUEBLA (MX) 2011-08-02 US disclosed
US-7989583-B2 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds BENEMERITA UNIVERSIDAD AUTONOMA DE PUEBLA (MX) 2011-08-02 US disclosed
US-7989583-B2 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds BENEMERITA UNIVERSIDAD AUTONOMA DE PUEBLA (MX) 2011-08-02 US disclosed
EP-2025697-A1 Process to obtain dimers, trimers and up to polymers from pyridinemethanol derivatives compounds Benemerita Universidad Autonoma de Puebla (MX) 2009-02-18 EP disclosed
EP-2025697-A1 Process to obtain dimers, trimers and up to polymers from pyridinemethanol derivatives compounds Benemerita Universidad Autonoma de Puebla (MX) 2009-02-18 EP disclosed
US-20090043063-A1 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds PERCINO ZACARIAS, Maria Judith (MX) 2009-02-12 US disclosed
US-20090043063-A1 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds PERCINO ZACARIAS, Maria Judith (MX) 2009-02-12 US disclosed
US-20090043063-A1 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds PERCINO ZACARIAS, Maria Judith (MX) 2009-02-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11718607-B2 Atypical coupling method for the preparation of 1,2-di(thiophen-2-yl)ethene-1,2-diol compounds via a Cu(II) catalyst AP2A2, AP2A1, DNM2 LMNA 4714/4885L3MBTL1 4181/4885P4HTM 4605/4885
US-10017474-B1 Method of synthesizing (E)-1,2-di(pyridin-2-yl) ethene-1,2-diol DPYSL2, DPYD, RER1 LMNA 1359/4885L3MBTL1 4225/4885P4HTM 786/4885
US-20090043063-A1 Process to obtain dimers, trimers and up to polymers from pyridinmethanol derivatives compounds PNPO, ADH1A, CYP2E1 LMNA 2020/4885L3MBTL1 4610/4885P4HTM 1009/4885
US-20220204487-A1 ATYPICAL COUPLING METHOD FOR THE PREPARATION OF 1,2-DI(THIOPHEN-2-YL)ETHENE-1,2-DIOL COMPOUNDS VIA A CU(II) CATALYST AP2A2, AP2A1, DNM2 LMNA 4714/4885L3MBTL1 4181/4885P4HTM 4605/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.