SCHEMBL2249558

SCHEMBL2249558

NC(=O)CC[C@H](NC(=O)c1ccc(-c2ccc3ccccc3c2)cc1)C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.58
CA1 P00915 2/20 0.58
PIN1 Q13526 3/20 0.53
UTS2R Q9UKP6 5/20 0.51
C3AR1 Q16581 1/20 0.51
MMP2 P08253 2/20 0.50
MMP9 P14780 2/20 0.50
MMP12 P39900 1/20 0.50
CTSL P07711 1/20 0.49
CTSB P07858 1/20 0.49
CTSS P25774 1/20 0.49
CTSK P43235 1/20 0.49
PTPN1 P18031 1/20 0.48
HPGDS O60760 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7407613 0.90 PIN1 (0.64) CA2CA1PIN1PTPN1
SCHEMBL2245325 0.90 CA2 (0.69) CA2CA1C3AR1MMP2MMP9
SCHEMBL2246061 0.90 CA2 (0.69) CA2CA1C3AR1MMP2MMP9
SCHEMBL2248592 0.86 DHFR (0.54) CA2CA1PIN1CTSLCTSB
SCHEMBL2249553 0.86 MMP12 (0.67) CA1UTS2RMMP12CTSLCTSB
SCHEMBL2248738 0.84 HPGDS (0.60) CA2CA1C3AR1MMP2MMP9
SCHEMBL5260684 0.83 CA2 (0.70) CA2CA1C3AR1MMP2MMP9
SCHEMBL5260686 0.83 CA2 (0.70) CA2CA1C3AR1MMP2MMP9
SCHEMBL2252396 0.82 CA2 (0.57) CA2CA1C3AR1MMP2MMP9
SCHEMBL2245609 0.82 CA2 (0.66) CA2CA1C3AR1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed