SCHEMBL2263014

SCHEMBL2263014

CCOC(=O)Cc1cnc2ccc(Br)cn12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
RXFP1 Q9HBX9 2/20 0.46
MAPT P10636 1/20 0.46
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
PSD A5PKW4 1/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
ADORA2A P29274 1/20 0.39
PIK3CA P42336 1/20 0.38
MTOR P42345 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TGFBR1 P36897 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28742005 0.87 KDM4E (0.43) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL2260441 0.84 KDM4E (0.47) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL23219125 0.83 TBXAS1 (0.45) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL29852848 0.83 TBXAS1 (0.45) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL3604567 0.83 TGFBR1 (0.43) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL2265835 0.82 TGFBR1 (0.43) KDM4ESMN1; SMN2RXFP1GLAGAA
SCHEMBL3595719 0.81 KDM4E (0.42) KDM4ESMN1; SMN2MAPTGLAGAA
SCHEMBL20985982 0.81 KDM4E (0.45) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL3595383 0.80 POLB (0.46) KDM4ESMN1; SMN2RXFP1MAPTGLA
SCHEMBL2261118 0.78 MAPK1 (0.49) KDM4ESMN1; SMN2RXFP1MAPTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250114345-A1 COMPOUNDS AND COMPOSITIONS AS CBP/P300 DEGRADERS AND USES THEREOF ONCOPIA THERAPEUTICS, INC. D/B/A/ SK LIFE SCIENCE LABS 2025-04-10 US disclosed
WO-2025049994-A1 COMPOUNDS AND COMPOSITIONS AS CBP/P300 DEGRADERS AND USES THEREOF ONCOPIA THERAPEUTICS, INC. D/B/A SK LIFE SCIENCE LABS (US) 2025-03-06 WO disclosed
US-20110294792-A1 PURINE DERIVATIVES AS KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2011-12-01 US disclosed
US-8058425-B2 Purine derivatives as kinase inhibitors ELI LILLY AND COMPANY (US) 2011-11-15 US disclosed
US-8022065-B2 Purine derivatives as kinase inhibitors ELI LILLY AND COMPANY (US) 2011-09-20 US disclosed
US-20110207721-A1 PURINE DERIVATIVES AS KINASE INHIBITORS ELI LILLY AND COMPANY (US) 2011-08-25 US disclosed
US-20090105229-A1 PURINE DERIVATIVES AS KINASE INHIBITORS ELI LILLY AND COMPANY 2009-04-23 US disclosed
US-7491716-B2 Purine derivatives as kinase inhibitors ELI LILLY AND COMPANY (US) 2009-02-17 US disclosed
US-7405299-B2 Compounds as pharmaceutical agents ELI LILLY AND COMPANY (US) 2008-07-29 US disclosed
EP-1483265-B1 PURINE DERIVATIVES AS KINASE INHIBITORS LILLY CO ELI (US) 2006-11-22 EP disclosed
US-20060058295-A1 Novel compounds as pharmaceutical agents ELI LILLY AND COMPANY (US) 2006-03-16 US disclosed
EP-1567527-A1 CONDENSED PYRAZOLO DERIVATIVES ELI LILLY AND COMPANY (US) 2005-08-31 EP disclosed
US-20050090483-A1 Purine derivatives as kinase inhibitors ELI LILLY AND COMPANY 2005-04-28 US disclosed
WO-2004050659-A1 NOVEL COMPOUNDS AS PHARMACEUTICAL AGENTS ELI LILLY AND COMPANY (US) 2004-06-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060058295-A1 Novel compounds as pharmaceutical agents TGFB1, TGFB2, TGFBR1 KDM4E 4107/4885SMN1; SMN2 2545/4885RXFP1 435/4885
US-20050090483-A1 Purine derivatives as kinase inhibitors PNP, ADK, NME2 KDM4E 1308/4885SMN1; SMN2 4465/4885RXFP1 2572/4885
US-20110294792-A1 PURINE DERIVATIVES AS KINASE INHIBITORS PNP, ADK, NME2 KDM4E 1308/4885SMN1; SMN2 4465/4885RXFP1 2572/4885
US-20110207721-A1 PURINE DERIVATIVES AS KINASE INHIBITORS PNP, ADK, NME2 KDM4E 1308/4885SMN1; SMN2 4465/4885RXFP1 2572/4885
US-20250114345-A1 COMPOUNDS AND COMPOSITIONS AS CBP/P300 DEGRADERS AND USES THEREOF EP300, CREBBP, HDAC1 KDM4E 200/4885SMN1; SMN2 3372/4885RXFP1 2455/4885
US-20090105229-A1 PURINE DERIVATIVES AS KINASE INHIBITORS PNP, ADK, NME2 KDM4E 1308/4885SMN1; SMN2 4465/4885RXFP1 2572/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.