SCHEMBL22650599

SCHEMBL22650599

Cc1nn2ccc(-c3ccnc(Nc4ccc(S(N)(=O)=O)nc4)n3)cc2c1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 2/20 0.43
GSK3B P49841 2/20 0.43
SMG1 Q96Q15 6/20 0.42
MTOR P42345 7/20 0.41
CDK1 P06493 7/20 0.40
IKBKB O14920 6/20 0.40
CDK2 P24941 6/20 0.40
MAPK8 P45983 1/20 0.39
MAPK10 P53779 1/20 0.39
CDK4 P11802 2/20 0.39
CCNB1 P14635 2/20 0.39
CCND1 P24385 1/20 0.39
PIK3CA P42336 1/20 0.38
PIK3CG P48736 1/20 0.38
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650701 0.74 JAK2 (0.38) GSK3BCDK1CDK2MAPK8MAPK10
SCHEMBL22650918 0.73 DKK1 (0.57) DKK1GSK3BSMG1MTORCDK1
SCHEMBL22650716 0.73 JAK2 (0.38) CDK1MAPK8MAPK10CDK4CCNB1
SCHEMBL22650604 0.72 JAK2 (0.37) SMG1CDK1MAPK8MAPK10CDK4
SCHEMBL22650423 0.72 JAK2 (0.37) GSK3BCDK1IKBKBCDK2MAPK8
SCHEMBL22650930 0.69 CDK4 (0.50) CDK1CDK2CDK4CCNB1CCND1
SCHEMBL22650923 0.66 MAPK8 (0.54) GSK3BCDK1IKBKBCDK2MAPK8
SCHEMBL22650920 0.64 CDK2 (0.54) CDK1CDK2MAPK8MAPK10CDK4
SCHEMBL22650919 0.63 CDK2 (0.54) GSK3BCDK1CDK2MAPK8MAPK10
SCHEMBL3517290 0.63 IKBKB (0.78) DKK1GSK3BCDK1IKBKBCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed