SCHEMBL22650910

SCHEMBL22650910

CCCN(C)C1CCN(c2ccc(N)nc2)C(=O)C1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.35
DRD2 P14416 8/20 0.35
DRD4 P21917 6/20 0.34
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
AKR1C3 P42330 1/20 0.32
HTR1A P08908 1/20 0.32
HTR1D P28221 1/20 0.32
PIK3CA P42336 1/20 0.32
MTOR P42345 1/20 0.32
CHIT1 Q13231 1/20 0.31
CHIA Q9BZP6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650566 0.90 DPP4 (0.33) AKR1C3PIK3CAMTOR
SCHEMBL22650368 0.85 ALOX5AP (0.37) AKR1C3PIK3CAMTOR
SCHEMBL29462389 0.85 ALOX5AP (0.37) AKR1C3PIK3CAMTOR
SCHEMBL22650562 0.84 PIK3CA (0.35) DRD3DRD2DRD4AKR1C3PIK3CA
SCHEMBL29491165 0.76 SPR (0.38) ROCK2PIK3CA
SCHEMBL22650412 0.76 SPR (0.38) ROCK2PIK3CA
SCHEMBL22650571 0.76 CCR5 (0.39) ROCK2
SCHEMBL22650730 0.73 ALOX5AP (0.40) AKR1C3PIK3CAMTOR
SCHEMBL25949319 0.73 DRD3 (0.43) DRD3DRD2DRD4
SCHEMBL13768888 0.71 CDK4 (0.46) PIK3CAMTORCHIT1CHIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021226140-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2021-11-11 WO disclosed
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed