SCHEMBL22650571

SCHEMBL22650571

CCN(C(=O)OC(C)(C)C)C1CCN(c2ccc(N)nc2)C(=O)C1

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.39
GPR119 Q8TDV5 16/20 0.37
SCN9A Q15858 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
ROCK2 O75116 1/20 0.34
LIPE Q05469 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650573 0.89 LIPE (0.35) GPR119SCN9ASCN10AROCK2LIPE
SCHEMBL22650412 0.87 SPR (0.38) GPR119ROCK2
SCHEMBL29491165 0.87 SPR (0.38) GPR119ROCK2
SCHEMBL22650572 0.81 CCR5 (0.38) CCR5GPR119LIPE
SCHEMBL22650562 0.81 PIK3CA (0.35)
SCHEMBL29462389 0.77 ALOX5AP (0.37)
SCHEMBL22650368 0.77 ALOX5AP (0.37)
SCHEMBL22650570 0.76 LIPE (0.37) CCR5GPR119ROCK2LIPE
SCHEMBL22650910 0.76 DRD3 (0.35) ROCK2
SCHEMBL18291712 0.75 CKS1B (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed