SCHEMBL22659705

SCHEMBL22659705

O=S(=O)(Cl)c1ccccc1-c1cncc2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 13/20 0.45
PRKCZ Q05513 1/20 0.45
CYP11B2 P19099 5/20 0.43
CYP11B1 P15538 3/20 0.43
CYP3A4 P08684 1/20 0.43
SLC22A12 Q96S37 1/20 0.42
KCNA5 P22460 1/20 0.41
KCNH2 Q12809 1/20 0.41
ERN1 O75460 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3909203 0.83 CA1 (0.52)
SCHEMBL3063215 0.81 CA1 (0.41) CYP17A1PRKCZCYP3A4
SCHEMBL20873066 0.78 PRKCZ (0.64) CYP17A1PRKCZCYP11B2CYP11B1CYP3A4
SCHEMBL7127239 0.76 ALDH1A1 (0.48)
SCHEMBL28481339 0.76 ROCK2 (0.41) PRKCZCYP3A4KCNH2
SCHEMBL27329478 0.72 CYP11B1 (0.53) CYP17A1PRKCZCYP11B2CYP11B1CYP3A4
SCHEMBL115053 0.71 CYP3A4 (0.56) PRKCZCYP3A4KCNH2
SCHEMBL29546384 0.71 CYP3A4 (0.56) PRKCZCYP3A4KCNH2
SCHEMBL10094643 0.70 CYP11B2 (0.54) CYP17A1PRKCZCYP11B2CYP11B1CYP3A4
SCHEMBL5617403 0.70 CYP11B2 (0.53) CYP17A1PRKCZCYP11B2CYP11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3921308-A1 SODIUM-HYDROGEN EXCHANGER 3 INHIBITOR COMPOUNDS ELI LILLY AND COMPANY (US) 2021-12-15 EP disclosed
WO-2020231770-A1 SODIUM-HYDROGEN EXCHANGER 3 INHIBITOR COMPOUNDS ELI LILLY AND COMPANY (US) 2020-11-19 WO disclosed