SCHEMBL22685248

SCHEMBL22685248

COc1ccc(C(=O)NC2(c3ccc(-c4ccc(C(F)(F)F)nc4N)cc3)CC2)cn1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.39
ROCK2 O75116 2/20 0.38
ROCK1 Q13464 2/20 0.38
NNMT P40261 1/20 0.37
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
EGLN1 Q9GZT9 2/20 0.37
BTK Q06187 1/20 0.36
KCNH2 Q12809 3/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PIK3CA P42336 2/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
PDE2A O00408 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22685244 0.92 WDR91 (0.40) PTPN1NNMTMKNK1MKNK2KCNH2
SCHEMBL22685250 0.86 PTPN1 (0.40) PTPN1ROCK2ROCK1NNMTMKNK1
SCHEMBL22684799 0.84 IDO1 (0.39) KCNH2HDAC3HDAC1HDAC2HDAC6
SCHEMBL22685330 0.80 CXCR3 (0.42) EGLN1PDE2A
SCHEMBL22685173 0.79 IDO1 (0.42) PDE2A
SCHEMBL22686783 0.79 WDR91 (0.42) ROCK2ROCK1BTKKCNH2HDAC3
SCHEMBL22685247 0.77 ROCK2 (0.41) PTPN1ROCK2ROCK1HDAC3HDAC1
SCHEMBL22685327 0.76 PDE2A (0.39) PDE2A
SCHEMBL22685191 0.76 WDR91 (0.43) KCNH2PDE2A
SCHEMBL22685351 0.75 WDR91 (0.54) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020228823-A1 NOVEL AMIDE COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2020-11-19 WO disclosed