SCHEMBL22747872

SCHEMBL22747872

O=C(O)c1c(C2CNCCO2)c2cc(Cl)c(Br)cc2n1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28556217 0.88 ALDH1A1 (0.43)
SCHEMBL22747834 0.79 KCNH2 (0.39) KCNH2TAAR1DRD2HTR2A
SCHEMBL22747875 0.79 EDNRA (0.36)
SCHEMBL22747877 0.76 KCNH2 (0.38) KCNH2TAAR1DRD2HTR2A
SCHEMBL22747873 0.72 MAT2A (0.43)
SCHEMBL28912331 0.69 FOLH1 (0.37)
SCHEMBL22760046 0.69 REN (0.38)
SCHEMBL22760356 0.68 MAT2A (0.43)
SCHEMBL22747849 0.67 FOLH1 (0.39)
SCHEMBL22760096 0.67 REN (0.39) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020244462-A1 INDOLE DERIVATIVES AND PHARMACEUTICAL USE THEREOF 中国药科大学 2020-12-10 WO disclosed
CN-112028815-A Indole derivatives and medical application thereof 中国药科大学 2020-12-04 CN disclosed