SCHEMBL22925622

SCHEMBL22925622

N#Cc1ccc(Nc2cc(-c3ccc(C(F)(F)F)cc3)no2)cn1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.41
CHEK1 O14757 14/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
CSGALNACT1 Q8TDX6 1/20 0.38
CDK2 P24941 1/20 0.37
AKT1 P31749 1/20 0.37
USP30 Q70CQ3 1/20 0.37
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22926103 0.88 CHEK1 (0.38) DGAT1CHEK1
SCHEMBL29620922 0.88 CHEK1 (0.38) DGAT1CHEK1
SCHEMBL22925913 0.77 HDAC6 (0.43) DGAT1CHEK1
SCHEMBL29620964 0.77 HSD11B1 (0.45) DGAT1CHEK1
SCHEMBL24636908 0.77 HSD11B1 (0.45) DGAT1CHEK1
SCHEMBL22925623 0.76 ACR (0.40) CYP3A4CYP2C19CSGALNACT1CDK2AKT1
SCHEMBL28733616 0.76 ACR (0.40) CYP3A4CYP2C19CSGALNACT1CDK2AKT1
SCHEMBL22926105 0.76 LRRK2 (0.40) DGAT1CHEK1
SCHEMBL22925496 0.74 TRPV1 (0.47) CHEK1
SCHEMBL29620971 0.74 GSK3B (0.62) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114450281-B Inhibitor compounds 辛塞拉治疗私人有限公司 2024-08-16 CN disclosed
US-20220274970-A1 INHIBITOR COMPOUNDS Cincera Therapeutics Pty Ltd (AU) 2022-09-01 US disclosed
EP-4003986-A1 INHIBITOR COMPOUNDS Cincera Therapeutics Pty Ltd (AU) 2022-06-01 EP disclosed
CN-114450281-A Inhibitor compounds 辛塞拉治疗私人有限公司 2022-05-06 CN disclosed
WO-2021012018-A1 INHIBITOR COMPOUNDS Cincera Therapeutics Pty Ltd (AU) 2021-01-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220274970-A1 INHIBITOR COMPOUNDS SERPINB1, MMP1, SSB DGAT1 164/4885CHEK1 1509/4885CYP3A4 4181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.