SCHEMBL2301546

SCHEMBL2301546

COc1cc(OC)cc(-c2cc(N3CCNC3=O)ccc2S(N)(=O)=O)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACVR1 Q04771 7/20 0.40
TGFBR1 P36897 2/20 0.40
RIPK2 O43353 5/20 0.38
NOD2 Q9HC29 5/20 0.38
CYP1A1 P04798 2/20 0.36
TNF P01375 1/20 0.36
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA4 P22748 2/20 0.36
CA7 P43166 2/20 0.36
SUV39H2 Q9H5I1 1/20 0.36
ADRB1 P08588 1/20 0.35
EGFR P00533 1/20 0.35
ROS1 P08922 1/20 0.35
ALK Q9UM73 1/20 0.35
CA12 O43570 2/20 0.34
CA9 Q16790 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301153 0.91 CA1 (0.43) TGFBR1TNFCA1CA2CA4
SCHEMBL2301613 0.90 TGFBR1 (0.42) ACVR1TGFBR1TNFCA1CA2
SCHEMBL2302730 0.89 ACVR1 (0.38) ACVR1TGFBR1RIPK2NOD2CYP1A1
SCHEMBL2303589 0.87 ACVR1 (0.43) ACVR1TGFBR1RIPK2CYP1A1CA1
SCHEMBL2301941 0.85 KDM4E (0.36) ACVR1CA1CA2SUV39H2CA12
SCHEMBL2304629 0.84 CA1 (0.47) ACVR1TGFBR1CA1CA2CA4
SCHEMBL2300277 0.83 CA12 (0.36) ACVR1CA1CA2SUV39H2EGFR
SCHEMBL2237662 0.82 PTGS2 (0.37) CA1CA2CA12CA9
SCHEMBL2299883 0.82 EIF2AK2 (0.41) CA1CA2EGFRROS1ALK
SCHEMBL2300517 0.81 PTGS2 (0.41) CA1CA2CA4CA7CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536693-A1 SUBSTITUTED 2-IMIDAZOLIDONES AND ANALOGS Université Laval (CA) 2012-12-26 EP disclosed
WO-2011100840-A1 SUBSTITUTED 2-IMIDAZOLIDONES AND ANALOGS UNIVERSITé LAVAL (CA) 2011-08-25 WO disclosed