SCHEMBL23218151

SCHEMBL23218151

OCc1c(-c2ccc(F)cc2)oc2ccc(Br)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 4/20 0.51
GABRD O14764 4/20 0.51
GABRA1 P14867 4/20 0.51
GABRB1 P18505 4/20 0.51
GABRG2 P18507 4/20 0.51
GABRB3 P28472 4/20 0.51
GABRA5 P31644 4/20 0.51
GABRA3 P34903 4/20 0.51
GABRA2 P47869 4/20 0.51
GABRB2 P47870 4/20 0.51
GABRA4 P48169 4/20 0.51
GABRE P78334 4/20 0.51
GABRA6 Q16445 4/20 0.51
GABRG1 Q8N1C3 4/20 0.51
GABRG3 Q99928 4/20 0.51
GABRQ Q9UN88 4/20 0.51
KMT2A Q03164 1/20 0.39
ANO1 Q5XXA6 4/20 0.38
PIM1 P11309 1/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29592241 1.00 GABRP (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL23218349 0.80 PIM1 (0.49) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29853136 0.72 KCNH2 (0.47) KMT2APIM1LMNASMN1; SMN2KCNH2
SCHEMBL23218435 0.72 KCNH2 (0.47) KMT2APIM1LMNASMN1; SMN2KCNH2
SCHEMBL2401078 0.72 ALOX5 (0.65) KMT2AKDM4E
SCHEMBL2404910 0.72 ATM (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL29852823 0.72 ATM (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL14764491 0.72 CYP3A4 (0.51) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL28159082 0.71 MEN1 (0.48) KMT2AANO1KDM4ELMNASMN1; SMN2
SCHEMBL23218086 0.70 PIM1 (0.45) KMT2APIM1LMNAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12558341-B2 Oral complement factor D inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2026-02-24 US disclosed
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-06-12 US disclosed
EP-4041238-A1 ORAL COMPLEMENT FACTOR D INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-08-17 EP disclosed
CN-114502168-A Oral complement factor D inhibitors 拜奥克里斯特制药公司 2022-05-13 CN disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
US-20160361275-A1 SUBSTITUTED PHENETHYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY ACADIA PHARMACEUTICALS INC. 2016-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160361275-A1 SUBSTITUTED PHENETHYLAMINES WITH SEROTONINERGIC AND/OR NOREPINEPHRINERGIC ACTIVITY SLC6A4, HTR4, GPR34 GABRP 110/4885GABRD 1347/4885GABRA1 649/4885
US-12558341-B2 Oral complement factor D inhibitors CFD, CFH, CFB GABRP 2631/4885GABRD 2643/4885GABRA1 3792/4885
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS CFD, CFH, CFB GABRP 3568/4885GABRD 3702/4885GABRA1 4487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.