SCHEMBL2324749

SCHEMBL2324749

COc1cccc(-c2oc(-c3nn(Cc4nc(C(C)=O)cs4)nc3C(N)=O)nc2C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.46
ADORA2A P29274 1/20 0.39
KMT2A Q03164 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
LDHA P00338 2/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
LMNA P02545 2/20 0.35
GPR35 Q9HC97 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PTGER1 P34995 1/20 0.35
PIN1 Q13526 1/20 0.35
CSNK2A1 P68400 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2326938 0.92 LDHA (0.39) IKBKBADORA2ALDHAIRAK4PTGER1
SCHEMBL2334798 0.89 PTGER1 (0.39) IKBKBADORA2ALDHAKDM4EHSD17B10
SCHEMBL2328798 0.89 PTGER1 (0.38) IKBKBADORA2ALDHAALDH1A1KDM4E
SCHEMBL2329257 0.89 IKBKB (0.43) IKBKBADORA2AKMT2ARXRARXRB
SCHEMBL1704018 0.88 IKBKB (0.43) IKBKBADORA2AKMT2ARXRARXRB
SCHEMBL2327504 0.87 PTGER1 (0.38) IKBKBADORA2APTGER1CSNK2A1SMN1; SMN2
SCHEMBL2324316 0.85 IKBKB (0.47) IKBKBADORA2AKMT2ARXRARXRB
SCHEMBL2327049 0.84 IKBKB (0.48) IKBKBADORA2AKMT2ARXRARXRB
SCHEMBL2332145 0.83 MMP1 (0.38) IKBKBLDHAALDH1A1HPGDKDM4E
SCHEMBL1704159 0.79 IKBKB (0.44) IKBKBADORA2AKMT2ARXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP claimed