SCHEMBL2330747

SCHEMBL2330747

CC(=O)c1ccc(Cn2nc(C(N)=O)c(-c3nc(C(=O)O)c(-c4cccc(Cl)c4)o3)n2)s1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.44
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RXRG P48443 2/20 0.35
NR4A2 P43354 1/20 0.35
SLC9A1 P19634 1/20 0.35
MDM2 Q00987 4/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PIN1 Q13526 1/20 0.34
ADORA2A P29274 1/20 0.33
PTPN11 Q06124 1/20 0.33
KDR P35968 1/20 0.33
PTGER1 P34995 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2331129 0.91 RXRA (0.36) IKBKBKMT2AMEN1RXRARXRB
SCHEMBL2324582 0.90 IKBKB (0.39) IKBKBPOLBKMT2AMEN1NR4A2
SCHEMBL2327822 0.90 TRPM8 (0.36) IKBKBSMN1; SMN2SLC9A1PIN1ADORA2A
SCHEMBL2324316 0.89 IKBKB (0.47) IKBKBNPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL2332003 0.89 FYN (0.39) IKBKBSMN1; SMN2ADORA2A
SCHEMBL2330683 0.86 ADORA2A (0.38) IKBKBADORA2A
SCHEMBL2331664 0.84 MAPK14 (0.34) IKBKB
SCHEMBL2329257 0.84 IKBKB (0.43) IKBKBNPC1RAB9AKMT2AMEN1
SCHEMBL2331266 0.84 IKBKB (0.45) IKBKBRAB9AKMT2AMEN1RXRA
SCHEMBL1704456 0.81 IKBKB (0.41) IKBKBNPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP claimed
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP disclosed