SCHEMBL2332003

SCHEMBL2332003

CC(=O)c1ccc(Cn2nc(C(N)=O)c(-c3nc(C(=O)O)c(-c4cccc(N(C)C)c4)o3)n2)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.34
LRRK2 Q5S007 1/20 0.34
HSD17B1 P14061 2/20 0.33
HSD17B2 P37059 2/20 0.33
ADORA2A P29274 1/20 0.33
GPR52 Q9Y2T5 1/20 0.32
IKBKB O14920 3/20 0.32
TRPM8 Q7Z2W7 1/20 0.32
CDK4 P11802 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCND3 P30281 1/20 0.31
CDK6 Q00534 1/20 0.31
ITK Q08881 1/20 0.31
CSNK2A1 P68400 1/20 0.30
NOTUM Q6P988 1/20 0.30
KDM4E B2RXH2 1/20 0.30
PPARG P37231 1/20 0.30
NCOA2 Q15596 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2331129 0.89 RXRA (0.36) HSD17B1HSD17B2ADORA2AIKBKBKDM4E
SCHEMBL2324582 0.89 IKBKB (0.39) ADORA2AIKBKBKDM4EPPARGNCOA2
SCHEMBL2330747 0.89 IKBKB (0.44) SMN1; SMN2ADORA2AIKBKB
SCHEMBL2327822 0.89 TRPM8 (0.36) SMN1; SMN2ADORA2AIKBKBTRPM8KDM4E
SCHEMBL2324316 0.87 IKBKB (0.47) SMN1; SMN2ADORA2AIKBKBKDM4EHSD17B10
SCHEMBL2330683 0.85 ADORA2A (0.38) FYNADORA2AIKBKBPPARGSLC16A3
SCHEMBL2327504 0.85 PTGER1 (0.38) FYNSMN1; SMN2LRRK2ADORA2AGPR52
SCHEMBL2327570 0.85 LRRK2 (0.36) FYNSMN1; SMN2LRRK2ADORA2AIKBKB
SCHEMBL2331664 0.83 MAPK14 (0.34) IKBKB
SCHEMBL1703783 0.82 LRRK2 (0.35) SMN1; SMN2LRRK2GPR52CSNK2A1SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP claimed
EP-2225231-B1 AMINOTRIAZOLE DERIVATIVES AS ALX AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2011-08-17 EP disclosed