SCHEMBL23536137

SCHEMBL23536137

Fc1cc(Cl)ccc1C1CCN(c2ccccc2I)CC1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 11/20 0.42
OPRL1 P41146 6/20 0.41
HTR1A P08908 1/20 0.38
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536100 0.84 MEN1 (0.49) GRM2OPRL1
SCHEMBL23536030 0.82 GRM2 (0.43) GRM2OPRL1
SCHEMBL23536314 0.82 GRM2 (0.43) GRM2OPRL1
SCHEMBL28867411 0.82 OPRL1 (0.42) GRM2OPRL1
SCHEMBL29932127 0.81 GRM2 (0.43) GRM2OPRL1
SCHEMBL23536378 0.81 GRM2 (0.43) GRM2OPRL1
SCHEMBL29931877 0.79 CA2 (0.43) GRM2OPRL1
SCHEMBL29931835 0.79 PGR (0.36) OPRL1
SCHEMBL23536154 0.77 OPRL1 (0.42) GRM2OPRL1
SCHEMBL23536205 0.76 HTR1A (0.51) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4076423-A1 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2022-10-26 EP disclosed
CN-115087440-A TRPML modulators 卡斯玛治疗公司 2022-09-20 CN disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed