SCHEMBL2354020

SCHEMBL2354020

Cc1cc(N(C(=O)O)c2ccc(C#N)cc2)ccc1Br

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.36
NPC1 O15118 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MEP1B Q16820 1/20 0.34
CYP2A6 P11509 1/20 0.34
GSK3B P49841 2/20 0.34
RAB9A P51151 2/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CETP P11597 1/20 0.33
AR P10275 1/20 0.33
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2179019 0.82 MT-CO2 (0.35) CYP19A1GAAAR
SCHEMBL14698064 0.76 KMT2A (0.54) NPC1MEN1KMT2AALDH1A1RAB9A
SCHEMBL18625530 0.74 ALDH1A1 (0.45) MEN1KMT2AALDH1A1POLBGAA
SCHEMBL16584847 0.73 GSK3B (0.45) ALDH1A1CYP2A6GSK3BCA1CA2
SCHEMBL152218 0.72 ALDH1A1 (0.46) MEN1KMT2AALDH1A1CYP2A6CA2
SCHEMBL18556032 0.72 RAB9A (0.43) NPC1MEN1KMT2AALDH1A1RAB9A
SCHEMBL9394223 0.70 PKM (0.35) NPC1MEN1KMT2AALDH1A1RAB9A
SCHEMBL14697483 0.69 KCNA5 (0.46) NPC1MEN1KMT2AALDH1A1GSK3B
SCHEMBL1705319 0.69 CA2 (0.45) ALDH1A1CYP2A6GSK3BGAACA1
SCHEMBL3840073 0.68 MEN1 (0.42) NPC1MEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2348863-A1 BORON-CONTAINING SMALL MOLECULES Anacor Pharmaceuticals, Inc. (US) 2011-08-03 EP disclosed
WO-2010027975-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2010-03-11 WO disclosed