SCHEMBL2368787

SCHEMBL2368787

c1ccc(COc2ncc3c(-c4ccccc4)csc3n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.42
ALDH1A1 P00352 6/20 0.42
HSD17B10 Q99714 4/20 0.42
CYP2C9 P11712 4/20 0.42
CYP2C19 P33261 4/20 0.42
CYP3A4 P08684 3/20 0.42
CASP1 P29466 3/20 0.42
CASP7 P55210 3/20 0.42
PIN1 Q13526 1/20 0.41
TSHR P16473 3/20 0.40
CLK4 Q9HAZ1 2/20 0.40
PDE5A O76074 1/20 0.40
SQOR Q9Y6N5 1/20 0.39
ESR1 P03372 1/20 0.39
P2RY14 Q15391 1/20 0.39
HPGD P15428 2/20 0.38
MAPK1 P28482 2/20 0.38
IKBKB O14920 1/20 0.38
HIF1A Q16665 1/20 0.38
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2368984 0.81 FGFR1 (0.41) CYP1A2ALDH1A1HSD17B10TSHRCLK4
SCHEMBL6356763 0.81 SQOR (0.37) CYP1A2ALDH1A1HSD17B10CYP2C9CYP3A4
SCHEMBL6359949 0.77 SQOR (0.37) ALDH1A1CLK4PDE5ASQORESR1
SCHEMBL2368935 0.75 ALDH1A1 (0.44) CYP1A2ALDH1A1HSD17B10TSHRCLK4
SCHEMBL30341183 0.74 NPC1 (0.47) CYP1A2ALDH1A1CYP2C9CYP2C19CLK4
SCHEMBL2368300 0.73 ESR1 (0.47) CYP1A2ALDH1A1HSD17B10CYP2C9CYP2C19
SCHEMBL14965210 0.73 ADORA1 (0.50) ALDH1A1CLK4DAPK3PRKD3MAP4K4
SCHEMBL30341175 0.73 ALDH1A1 (0.46) CYP1A2ALDH1A1TSHRCLK4HPGD
SCHEMBL6358684 0.72 LMNA (0.40) ALDH1A1HSD17B10TSHRCLK4MAPK1
SCHEMBL2368759 0.71 BTK (0.39) ALDH1A1HSD17B10CASP7TSHRCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022076-B2 Thieno[2,3-d]pyrimidine derivatives as potassium channel modulators; antiarrhythmia agents XENTION LIMITED (GB) 2011-09-20 US disclosed