SCHEMBL2373128

SCHEMBL2373128

CCCOC1(c2cccc(C(F)(F)F)c2)C=C(C(N)=O)c2ccccc2N1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
ALDH1A1 P00352 2/20 0.33
EPHX1 P07099 2/20 0.33
USP2 O75604 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
KDR P35968 1/20 0.33
MAOB P27338 1/20 0.33
GALR3 O60755 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
POLB P06746 1/20 0.33
OPRM1 P35372 2/20 0.33
OPRL1 P41146 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2461669 0.78 HCAR3 (0.39) HCAR3HCAR2ALDH1A1KDRGALR3
SCHEMBL25329372 0.65 ALDH1A1 (0.38) ALDH1A1GALR3OPRM1OPRL1CACNA1F
SCHEMBL19691189 0.62 ALDH1A1 (0.41) ALDH1A1POLBMEN1KMT2ALMNA
Butane SCHEMBL27384864 0.61 ALDH1A1 (0.61) ALDH1A1EPHX1TAS1R3TAS1R1MAOB
SCHEMBL5045630 0.61 NOS2 (0.32) ALDH1A1POLBOPRM1
SCHEMBL31575815 0.59 LMNA (0.60) ALDH1A1USP2TAS1R3TAS1R1KDR
SCHEMBL20267329 0.59 LMNA (0.60) ALDH1A1USP2TAS1R3TAS1R1KDR
SCHEMBL15821917 0.58 CES2 (0.47) ALDH1A1EPHX1TAS1R3TAS1R1HDAC3
SCHEMBL14939165 0.57 MAPT (0.49) HCAR3HCAR2MAOBGALR3OPRM1
SCHEMBL13386454 0.57 KDM1A (0.51) HCAR3HCAR2HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119704-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed