SCHEMBL23770508

SCHEMBL23770508

CCOC(=O)C1(C)CCN(c2cccc(SNc3ccc(Cl)c(-c4cc(F)ccc4C)n3)n2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.35
RET P07949 3/20 0.32
DGAT2 Q96PD7 1/20 0.32
P2RY1 P47900 1/20 0.32
CNR1 P21554 1/20 0.32
OPRM1 P35372 2/20 0.32
CTSA P10619 1/20 0.32
SMO Q99835 1/20 0.32
P2RY12 Q9H244 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770864 0.90 HDAC3 (0.34) RETP2RY1CNR1OPRM1SMO
SCHEMBL23770853 0.90 ABL1 (0.34) ABL1RETOPRM1PTPN11JAK2
SCHEMBL23770789 0.88 HDAC3 (0.33) CNR1OPRM1CTSAHDAC3HDAC4
SCHEMBL23770829 0.87 HDAC3 (0.33) RETP2RY1CNR1OPRM1SMO
SCHEMBL23770855 0.85 ABL1 (0.32) ABL1SMOPTPN11
SCHEMBL19925055 0.85 ABL1 (0.33) ABL1DGAT2P2RY1CNR1OPRM1
SCHEMBL23770868 0.82 PTPN11 (0.37) ABL1RETCNR1PTPN11MEN1
SCHEMBL23770446 0.81 SUV39H2 (0.39) RETSMOMEN1KMT2A
SCHEMBL23770808 0.81 HTR3E (0.38) ABL1PTPN11
SCHEMBL23770757 0.81 MEN1 (0.33) OPRM1PTPN11JAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed