SCHEMBL23770668

SCHEMBL23770668

Cc1ccccc1-c1nc(NSc2cccc(N3CCCC(C(=O)O)C3)n2)ccc1Cl

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.40
P2RX7 Q99572 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HSD11B1 P28845 1/20 0.36
NOTUM Q6P988 3/20 0.36
SLC6A1 P30531 2/20 0.36
AKR1C3 P42330 2/20 0.35
MAP3K5 Q99683 1/20 0.35
AKR1C1 Q04828 1/20 0.35
MPL P40238 1/20 0.35
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770648 0.92 GPBAR1 (0.41) GPBAR1P2RX7KDM4EMEN1ALDH1A1
SCHEMBL23770656 0.90 P2RX7 (0.39) GPBAR1P2RX7KDM4EMEN1ALDH1A1
SCHEMBL23770813 0.90 ITGB2 (0.40) GPBAR1P2RX7KDM4EMEN1ALDH1A1
SCHEMBL23770485 0.89 P2RX7 (0.38) GPBAR1P2RX7KDM4EMEN1ALDH1A1
SCHEMBL23770488 0.88 ITGB2 (0.40) GPBAR1KDM4EMEN1ALDH1A1KMT2A
SCHEMBL23770759 0.84 MPL (0.43) GPBAR1P2RX7NOTUMAKR1C3AKR1C1
SCHEMBL23770608 0.83 NOTUM (0.41) NOTUMMPL
SCHEMBL23770893 0.82 GPBAR1 (0.39) GPBAR1KDM4EMEN1ALDH1A1KMT2A
SCHEMBL19970115 0.81 DGAT1 (0.34)
SCHEMBL23770806 0.80 RBP4 (0.36) NOTUMSLC6A1MPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed