SCHEMBL23770798

SCHEMBL23770798

OC1CN(c2cc(SNc3ccc(C(F)(F)F)c(-c4ccccc4C(F)(F)F)n3)ccn2)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 5/20 0.38
ICAM1 P05362 5/20 0.38
ITGAL P20701 5/20 0.38
CYP1A2 P05177 7/20 0.37
CYP2C19 P33261 4/20 0.37
CYP3A4 P08684 4/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 3/20 0.37
TSHR P16473 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP2D6 P10635 1/20 0.37
MPL P40238 1/20 0.36
SOS1 Q07889 1/20 0.35
CYP2C9 P11712 1/20 0.35
CLK2 P49760 1/20 0.34
LRRK2 Q5S007 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770583 0.86 RAF1 (0.36) ITGB2ICAM1ITGALMPLSOS1
SCHEMBL19951424 0.80 SCN9A (0.38) ITGB2ICAM1ITGALCYP1A2CYP2C19
SCHEMBL29464379 0.80 SCN9A (0.38) ITGB2ICAM1ITGALCYP1A2CYP2C19
SCHEMBL23770753 0.76 GRIN2B (0.36) MPLSOS1CLK2LRRK2PRKCA
SCHEMBL23770570 0.76 KRAS (0.33) LRRK2
SCHEMBL23770607 0.75 JAK2 (0.35) LRRK2
SCHEMBL19968862 0.74 SCN9A (0.37) ITGB2ICAM1ITGALMPLCLK2
SCHEMBL23770822 0.74 MPL (0.33) ALDH1A1MPLCLK2LRRK2PRKCA
SCHEMBL23770810 0.73 MPL (0.32) MPLPRKCAPRKCQPDE10A
SCHEMBL23770677 0.73 ABL1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed