SCHEMBL2408189

SCHEMBL2408189

CNC(=O)OC(c1cn(S(=O)(=O)c2cccc(-c3nnc(C)o3)c2)c(-c2cccnc2F)c1F)C(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR9 P51686 1/20 0.36
NAMPT P43490 1/20 0.35
CCKBR P32239 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
MAPK14 Q16539 1/20 0.31
LCLAT1 Q6UWP7 1/20 0.31
CTSV O60911 1/20 0.31
CTSL P07711 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
FGFR3 P22607 2/20 0.31
IDO1 P14902 1/20 0.31
MAPK1 P28482 1/20 0.31
KDR P35968 1/20 0.30
LMNA P02545 1/20 0.30
PTBP1 P26599 1/20 0.30
TYK2 P29597 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2408490 0.86 HTR6 (0.35)
SCHEMBL4425656 0.85 MET (0.39)
SCHEMBL2410027 0.83 NTRK1 (0.31)
SCHEMBL2414854 0.82 KDR (0.34) KDR
SCHEMBL5006275 0.82 CCR9 (0.35) CCR9NAMPTCCKBRLCLAT1
SCHEMBL1837632 0.81 PTGS2 (0.30)
SCHEMBL1831693 0.81
SCHEMBL1829458 0.81 RORC (0.32) NAMPT
SCHEMBL1832698 0.80 RORC (0.32) NAMPT
SCHEMBL2411543 0.80 ALDH1A1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed