SCHEMBL2409152

SCHEMBL2409152

CC(=O)c1cccc(S(=O)(=O)n2cc(CN(C)C(=O)OC(C)(C)C)cc2-c2cccnc2F)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CHRM5 P08912 1/20 0.34
KAT8 Q9H7Z6 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33
KAT6A Q92794 1/20 0.32
KAT5 Q92993 1/20 0.32
APAF1 O14727 1/20 0.32
UBE2N P61088 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CNR1 P21554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2409950 0.92 HTR6 (0.38) ALDH1A1KAT8HTR2CSLC6A4KAT6A
SCHEMBL31187457 0.90 KAT8 (0.35) KAT8PKMHTR2CSLC6A4KAT6A
SCHEMBL2415723 0.90 HTR2C (0.39) KAT8HTR2CSLC6A4KAT6AKAT5
SCHEMBL31187449 0.89 MET (0.42) ALDH1A1CHRM5PKMTSHR
SCHEMBL4418624 0.88 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2CHRM5GAAHTT
SCHEMBL1278111 0.88 RIPK1 (0.34) ALDH1A1SMN1; SMN2KAT8GAAPKM
SCHEMBL2412876 0.88 PTGDR2 (0.39) KAT8GAAHTR2CSLC6A4KAT6A
SCHEMBL2414740 0.88 HTR2C (0.37) KAT8NPSR1PKMHTR2CSLC6A4
SCHEMBL2414119 0.87 RORC (0.37) KAT8KAT6AKAT5
SCHEMBL2412420 0.86 GRM4 (0.38) KAT8HTR2CSLC6A4KAT6AKAT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed