SCHEMBL2409158

SCHEMBL2409158

CC(=O)c1cccc(S(=O)(=O)n2cc(CN(CC(C)(C)C)C(=O)O)cc2-c2cccnc2F)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CHRM5 P08912 2/20 0.34
LMNA P02545 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
TSHR P16473 1/20 0.33
CNR1 P21554 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2418769 0.92 HTR6 (0.37) ALDH1A1GAAHTTNPSR1CHRM5
SCHEMBL2415727 0.91 CHRM5 (0.37) ALDH1A1GAAHTTNPSR1SMN1; SMN2
SCHEMBL2412879 0.87 PTGDR2 (0.43) ALDH1A1GAACHRM5CNR1L3MBTL1
SCHEMBL1278112 0.87 PTGER2 (0.36) ALDH1A1GAASMN1; SMN2TSHRPKM
SCHEMBL4418624 0.87 ALDH1A1 (0.39) ALDH1A1GAAHTTNPSR1SMN1; SMN2
SCHEMBL2414742 0.87 PKM (0.35) ALDH1A1GAACHRM5CNR1L3MBTL1
SCHEMBL2414122 0.87 PPME1 (0.36) ALDH1A1
SCHEMBL2412424 0.86 PTGDR2 (0.39) ALDH1A1NPSR1SMN1; SMN2LMNACRHBP
SCHEMBL1278414 0.85 PTGDR2 (0.34) ALDH1A1CHRM5CNR1L3MBTL1
SCHEMBL2408624 0.85 L3MBTL1 (0.33) ALDH1A1NPSR1L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed