SCHEMBL2409332

SCHEMBL2409332

CC(C)(C)C(Cc1cn(-c2cccnc2F)cc1F)NC(=O)O

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.32
NAPRT Q6XQN6 1/20 0.32
CPB1 P15086 1/20 0.32
CPB2 Q96IY4 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
MMP13 P45452 1/20 0.32
SCN9A Q15858 2/20 0.31
SCN10A Q9Y5Y9 1/20 0.31
MYC P01106 1/20 0.31
SLC13A5 Q86YT5 1/20 0.31
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2411005 0.90 P2RX7 (0.35) CTSACPB1CPB2
SCHEMBL1830978 0.72 DYRK1A (0.35) NAPRTMMP2MMP9MMP8MMP13
SCHEMBL2409335 0.71 HTR2C (0.39) CACNA1G
SCHEMBL3700741 0.70 PTGDR2 (0.34) CTSAMMP2MMP9MMP8MMP13
SCHEMBL2192366 0.70 DCTPP1 (0.31) MMP2MMP9MMP8MMP13
SCHEMBL476324 0.69 COMT (0.35) MMP2MMP9MMP8MMP13
SCHEMBL2194609 0.69 MMP2 (0.30) MMP2MMP9MMP8MMP13
SCHEMBL2410511 0.69 ABCC9 (0.33) MMP2MMP9MMP8MMP13
SCHEMBL2412156 0.68 DCTPP1 (0.32) MMP2MMP9MMP8MMP13
SCHEMBL2407099 0.68 OPRM1 (0.32) MMP2MMP9MMP8MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed