SCHEMBL24112688

SCHEMBL24112688

C=CC(=O)NCc1ccccc1NC

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 3/20 0.45
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 6/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 1/20 0.38
ATM Q13315 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HPGD P15428 2/20 0.37
EGFR P00533 1/20 0.36
FLT3 P36888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL59858 0.84 TGM2 (0.55) TGM2GAAKMT2AALDH1A1CYP2C9
SCHEMBL397784 0.82 ALDH1A1 (0.53) TGM2GAAKMT2AALDH1A1KDM4E
SCHEMBL3250028 0.81 PSIP1 (0.45) TGM2GAAKMT2AALDH1A1KDM4E
SCHEMBL5082541 0.80 KMT2A (0.67) TGM2GAAKMT2AALDH1A1KDM4E
SCHEMBL17258879 0.80 ALDH1A1 (0.49) GAAKMT2ATMEM97SIGMAR1ALDH1A1
SCHEMBL8337546 0.80 SETDB1 (0.50) KMT2ATMEM97SIGMAR1ALDH1A1KDM4E
SCHEMBL2449430 0.78 TGM2 (0.53) TGM2GAAKMT2AALDH1A1CYP2C9
SCHEMBL410698 0.78 TSHR (0.52) TGM2GAAKMT2AALDH1A1TSHR
SCHEMBL16634646 0.77 TGM2 (0.45) TGM2GAAKMT2AALDH1A1CYP2C9
SCHEMBL3270305 0.77 TGM2 (0.42) TGM2GAAKMT2AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252339-A1 SUBSTITUTED PURINE-2,6-DIONE COMPOUNDS AS KRAS INHIBITORS ACCUTAR BIOTECHNOLOGY, INC. (US) 2021-12-16 WO disclosed